Synthesis and biological evaluation of (R)- and (S)-2-(phosphonomethyl)pentanedioic acids as inhibitors of glutamate carboxypeptidase II

Tetrahedron Asymmetry

Volumn 13, Issue 15, 2002, Pages 1609-1614

  Vitharana, Dilrukshi ^a   France, Jessica E ^a   Scarpetti, David ^a   Bonneville, George W ^a   Majer, Pavel ^a   Tsukamoto, Takashi ^a  

^a GUILFORD PHARMACEUTICALS INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

2 (HYDROXYPHOSPHINOYLMETHYL)PENTANEDIOIC ACID DIBENZYL ESTER; 2 (PHOSPHONOMETHYL)PENTANEDIOIC ACID; ALPHA METHYLBENZYLAMINE; CARBON; ENZYME INHIBITOR; ESTER DERIVATIVE; GAMMA GLUTAMYL HYDROLASE; GLUTARIC ACID DERIVATIVE; HYDROGEN; MENTHOL; PHOSPHINIC ACID DERIVATIVE; PHOSPHONIC ACID DERIVATIVE; UNCLASSIFIED DRUG; YOHIMBINE;

ARTICLE; ATOM; BRAIN; CATALYSIS; DRUG ACTIVITY; DRUG POTENCY; DRUG PURITY; DRUG SYNTHESIS; ENANTIOMER; ENZYME INHIBITION; OXIDATION; PHOSPHORUS NUCLEAR MAGNETIC RESONANCE; PRIORITY JOURNAL; RACEMIC MIXTURE; TISSUE CULTURE; X RAY CRYSTALLOGRAPHY;

EID: 0037077789     PISSN: 09574166     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0957-4166(02)00412-3     Document Type: Article

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