Novel N-{ω-[4-(2-methoxyphenyl)piperazin-1-YL]-ethyl}pyrid-2(1H)-ones with diversified 5-HT1A receptor activity

Polish Journal of Pharmacology

Volumn 54, Issue 6, 2002, Pages 641-646

  Paluchowska, Maria H ^a   Bugno, Ryszard ^a   Charakchieva Minol, Sijka ^a   Wesołowska, Anna ^a   Chojnacka Wójcik, Ewa ^a  

^a INSTITUTE OF PHARMACOLOGY   (Poland)

Author keywords

Arylpiperazine 5 HT1A receptor ligands; Functional 5 HT1A receptor activity; Pyrid 2(1H) one derivatives

Indexed keywords

2 DIPROPYLAMINO 8 HYDROXYTETRALIN; ALIPHATIC COMPOUND; CYCLOBUTANE DERIVATIVE; N [2 [4 (2 METHOXYPHENYL) 1 PIPERAZINYL]ETHYL] N (2 PYRIDYL)CYCLOHEXANECARBOXAMIDE; N [OMEGA [4 (2 METHOXYPHENYL)PIPERAZIN 1 YL]ETHYL]PYRID 2(1H) ONE DERIVATIVE; N TERT BUTYL 3 [4 (2 METHOXYPHENYL) 1 PIPERAZINYL] 2 PHENYLPROPIONAMIDE; POSTSYNAPTIC RECEPTOR; SEROTONIN 1A AGONIST; SEROTONIN 1A ANTAGONIST; SEROTONIN 1A RECEPTOR; SEROTONIN 2A RECEPTOR; UNCLASSIFIED DRUG;

ANIMAL BEHAVIOR; ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; BRAIN TISSUE; CONTROLLED STUDY; DRUG POTENCY; DRUG SELECTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; IN VITRO STUDY; IN VIVO STUDY; INDUCED HYPOTHERMIA; LIGAND BINDING; MALE; NONHUMAN; RECEPTOR AFFINITY; RECEPTOR INTRINSIC ACTIVITY; STRUCTURE ACTIVITY RELATION;

ANIMALS; BODY TEMPERATURE; MALE; MICE; PIPERAZINES; RATS; RATS, WISTAR; RECEPTORS, SEROTONIN; RECEPTORS, SEROTONIN, 5-HT1; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0036968059     PISSN: 12306002     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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