1,4-Benzoxazin-3(4H)-one derivatives and related compounds as 5-HT(1A) and 5-HT(2A) receptor ligands; The effect of the terminal amide fragment on the 5-HT(1A)/5-HT(2A) affinity and functional activity

Polish Journal of Pharmacology

Volumn 50, Issue 4-5, 1998, Pages 333-340

  Mokrosz, Maria J ^a   Kowalski, Piotr ^b   Kowalska, Teresa ^b   Majka, Zbigniew ^b   Duszyńska, Beata ^a   Charakchieva Minol, Sijka ^a   Szaro, Anna ^a   Tatarczyńska, Ewa ^a   Kłodzińska, Aleksandra ^a   Chojnacka Wójcik, Ewa ^a  

^a INSTITUTE OF PHARMACOLOGY   (Poland)

^b CRACOW UNIVERSITY OF TECHNOLOGY   (Poland)

Author keywords

1,4 Benzoxazin 3(4H) one derivatives; 5 HT(1A) and 5 HT(2A) antagonistic properties; 5 HT(1A) and 5 HT(2A) ligands

Indexed keywords

2 DIPROPYLAMINO 8 HYDROXYTETRALIN; AMIDE; BENZOXAZINONE DERIVATIVE; LIGAND; PSYCHOTROPIC AGENT; SEROTONIN 1A ANTAGONIST; SEROTONIN 1A RECEPTOR; SEROTONIN 2A ANTAGONIST; SEROTONIN 2A RECEPTOR;

ANIMAL EXPERIMENT; ARTICLE; CONTROLLED STUDY; HEAD TWITCH; INTRAPERITONEAL DRUG ADMINISTRATION; MALE; MOUSE; NONHUMAN; RADIOASSAY; RAT; RECEPTOR AFFINITY; STRUCTURE ACTIVITY RELATION; SUBCUTANEOUS DRUG ADMINISTRATION;

8-HYDROXY-2-(DI-N-PROPYLAMINO)TETRALIN; ANIMALS; BEHAVIOR, ANIMAL; BODY TEMPERATURE; BRAIN; CEREBRAL CORTEX; DRUG INTERACTIONS; HEAD MOVEMENTS; HIPPOCAMPUS; LIGANDS; LIP; MALE; MICE; MUSCLE SPASTICITY; OXAZINES; RATS; RECEPTOR, SEROTONIN, 5-HT2A; RECEPTORS, SEROTONIN; RECEPTORS, SEROTONIN, 5-HT1; RESERPINE; SEROTONIN ANTAGONISTS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 7844219851     PISSN: 12306002     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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