Thalassiolins A-C: New marine-derived inhibitors of HIV cDNA integrase

Bioorganic and Medicinal Chemistry

Volumn 10, Issue 11, 2002, Pages 3619-3625

  Rowley, David C ^a,d   Hansen, Mark S T ^b   Rhodes, Denise ^b   Sotriffer, Christoph A ^c   Ni, Haihong ^c   McCammon, J Andrew ^c   Bushman, Frederic D ^b   Fenical, William ^a  

^a UNIVERSITY OF CALIFORNIA SAN DIEGO   (United States)

^b SALK INSTITUTE FOR BIOLOGICAL STUDIES   (United States)

^c San Diego   (United States)

^d UNIVERSITY OF RHODE ISLAND   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

BETA GLUCOSE; GLUCOSE DERIVATIVE; INTEGRASE; INTEGRASE INHIBITOR; THALASSIOLIN A; THALASSIOLIN B; THALASSIOLIN C; UNCLASSIFIED DRUG;

ARTICLE; BINDING SITE; BIOCHEMISTRY; CATALYST; CONTROLLED STUDY; CRYSTAL STRUCTURE; DRUG ISOLATION; DRUG POTENCY; ENZYME INHIBITION; HUMAN; HUMAN CELL; HUMAN IMMUNODEFICIENCY VIRUS 1; IC 50; MOLECULAR MODEL; MOLLUSCIPOXVIRUS; NONHUMAN; SEAGRASS; VIRUS REPLICATION;

BINDING SITES; CELLS, CULTURED; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; DNA, COMPLEMENTARY; FLAVONOIDS; HIV INFECTIONS; HIV INTEGRASE; HIV INTEGRASE INHIBITORS; HIV-1; HUMANS; HYDROCHARITACEAE; INDICATORS AND REAGENTS; MAGNETIC RESONANCE SPECTROSCOPY; MODELS, MOLECULAR; MOLECULAR CONFORMATION; SPECTROMETRY, MASS, MATRIX-ASSISTED LASER DESORPTION-IONIZATION;

HUMAN IMMUNODEFICIENCY VIRUS; HUMAN IMMUNODEFICIENCY VIRUS 1; THALASSIA; THALASSIA TESTUDINUM;

EID: 0036836956     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0968-0896(02)00241-9     Document Type: Article

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