Local injection of a selective endothelin-B receptor agonist inhibits endothelin-1-induced pain-like behavior and excitation of nociceptors in a naloxone-sensitive manner

Journal of Neuroscience

Volumn 22, Issue 17, 2002, Pages 7788-7796

  Khodorova, Alia ^a   Fareed, Moin U ^a   Gokin, Alexander ^a   Strichartz, Gary R ^a   Davar, Gudarz ^a,b  

^a HARVARD MEDICAL SCHOOL   (United States)

^b BRIGHAM AND WOMEN S HOSPITAL   (United States)

Author keywords

Analgesia; Endothelin 1; G protein; Nociception; Opioid; Potassium channel

Indexed keywords

ENDOTHELIN 1; ENDOTHELIN A RECEPTOR; ENDOTHELIN B RECEPTOR; ENDOTHELIN B RECEPTOR AGONIST; ENDOTHELIN B RECEPTOR ANTAGONIST; N (2,6 DIMETHYLPIPERIDINOCARBONYL) 4 METHYLLEUCYL DEXTRO (1 METHOXYCARBONYLTRYPTOPHANYL) DEXTRO NORLEUCINE; NALOXONE; OPIATE ANTAGONIST; SUCCINYLENDOTHELIN 1 [8-21][9 GLUTAMIC ACID 11,15 ALANINE];

ANIMAL EXPERIMENT; ARTICLE; CONTROLLED STUDY; MALE; NERVE CELL EXCITABILITY; NERVE ENDING; NERVE FIBER C; NEUROMODULATION; NOCICEPTION; NOCICEPTIVE RECEPTOR; NONHUMAN; PAIN; PRIORITY JOURNAL; RAT; RECEPTOR UPREGULATION; SIGNAL TRANSDUCTION; SPIKE;

EID: 0036758643     PISSN: 02706474     EISSN: None     Source Type: Journal    
DOI: 10.1523/jneurosci.22-17-07788.2002     Document Type: Article

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