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Volumn 45, Issue 16, 2002, Pages 3418-3429

Monocyclic human tachykinin NK-2 receptor antagonists as evolution of a potent bicyclic antagonist: QSAR and site-directed mutagenesis studies

(9) Giolitti, Alessandro a Altamura, Maria a Bellucci, Francesca a Giannotti, Danilo a Meini, Stefania a Patacchini, Riccardo a Rotondaro, Luigi a Zappitelli, Sabrina a Maggi, Carlo A a

a Menarini Ricerche SpA (Italy)

Author keywords

[No Author keywords available]

Indexed keywords

MEN 11523; MEN 11532; MEN 11540; MEN 11558; MEN 11667; MEN 11668; MEN 11690; MEN 11691; MEN 11701; MEN 11703; MEN 11708; MEN 11712; MEN 11715; MEN 11716; MEN 11733; MEN 11749; MEN 11755; MEN 11757; MEN 11799; MEN 11830; MEN 11842; MEN 11877; MEN 11959; MEN 11970; MEN 11983; MEN 11986; MEN 11987; NEUROKININ 2 RECEPTOR; NEUROKININ 2 RECEPTOR ANTAGONIST; TACHYKININ RECEPTOR ANTAGONIST; UNCLASSIFIED DRUG; UNINDEXED DRUG;

ARTICLE; DRUG BINDING SITE; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; MOLECULAR MODEL; POINT MUTATION; QUANTITATIVE STRUCTURE ACTIVITY RELATION; RECEPTOR AFFINITY; SITE DIRECTED MUTAGENESIS;

AMINO ACID SEQUENCE; BINDING SITES; BINDING, COMPETITIVE; HUMANS; LIGANDS; MODELS, MOLECULAR; MOLECULAR CONFORMATION; MOLECULAR MIMICRY; MOLECULAR SEQUENCE DATA; MUTAGENESIS, SITE-DIRECTED; PEPTIDES, CYCLIC; QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP; RADIOLIGAND ASSAY; RECEPTORS, NEUROKININ-2; TACHYKININS;

EID: 0036682427 PISSN: 00222623 EISSN: None Source Type: Journal
DOI: 10.1021/jm011127h Document Type: Article

Times cited : (14)

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* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.