MEN 11420 (Nepadutant), a novel glycosylated bicyclic peptide tachykinin NK2 receptor antagonist

British Journal of Pharmacology

Volumn 123, Issue 1, 1998, Pages 81-91

  Catalioto, R M ^a   Criscuoli, M ^a   Cucchi, P ^a   Giachetti, A ^a   Giannotti, D ^a   Giuliani, S ^a   Lecci, A ^a   Lippi, A ^a   Patacchini, R ^a   Quartara, L ^a   Renzetti, A R ^a   Tramontana, M ^a   Arcamone, F ^a   Maggi, C A ^a  

^a Menarini Ricerche SpA   (Italy)

Author keywords

MEN 11420; Neurokinin A; Receptors; Tachykinin NK2; Tachykinins

Indexed keywords

IODINE 125; ION CHANNEL; MEN 10627; NEPADUTANT; NEUROKININ 1 RECEPTOR; NEUROKININ 2 RECEPTOR; NEUROKININ 2 RECEPTOR ANTAGONIST; NEUROKININ 3 RECEPTOR; NEUROKININ A; SAREDUTANT; SUBSTANCE P SULFONE [9 PROLINE]; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANIMAL MODEL; ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; BLADDER; CONTROLLED STUDY; GUINEA PIG; HAMSTER; ILEUM; INTRADUODENAL DRUG ADMINISTRATION; INTRANASAL DRUG ADMINISTRATION; INTRAVENOUS DRUG ADMINISTRATION; MOUSE; NONHUMAN; PATHOPHYSIOLOGY; PORTAL VEIN; PRIORITY JOURNAL; PULMONARY ARTERY; RABBIT; RAT; RECEPTOR AFFINITY; RECTAL DRUG ADMINISTRATION; SMOOTH MUSCLE CONTRACTION; TRACHEA;

ANIMALS; CHO CELLS; CRICETINAE; FEMALE; GUINEA PIGS; HUMANS; ION CHANNELS; MALE; PEPTIDES, CYCLIC; RABBITS; RADIOLIGAND ASSAY; RATS; RATS, WISTAR; RECEPTORS, NEUROKININ-1; RECEPTORS, NEUROKININ-2; RECEPTORS, NEUROKININ-3;

EID: 6844266263     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0701587     Document Type: Article

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