Novel retinoid X receptor antagonists: Specific inhibition of retinoid synergism in RXR-RAR heterodimer actions

Journal of Medicinal Chemistry

Volumn 45, Issue 16, 2002, Pages 3327-3330

  Takahashi, Bitoku ^a   Ohta, Kiminori ^a   Kawachi, Emiko ^a   Fukasawa, Hiroshi ^a   Hashimoto, Yuichi ^a   Kagechika, Hiroyuki ^a  

^a UNIVERSITY OF TOKYO   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

2 AMINOPYRIMIDINE 5 CARBOXYLIC ACID DERIVATIVE; DIMER; PA 024; PYRIMIDINE DERIVATIVE; RECEPTOR BLOCKING AGENT; RETINOIC ACID RECEPTOR; RETINOID; RETINOID X RECEPTOR; TAMIBAROTENE; UNCLASSIFIED DRUG;

ARTICLE; BINDING SITE; CELL DIFFERENTIATION; CELL STRAIN HL 60; DRUG ANTAGONISM; DRUG POTENTIATION; HUMAN; HUMAN CELL; STRUCTURE ACTIVITY RELATION;

BENZOATES; CARBOXYLIC ACIDS; CELL DIFFERENTIATION; DEPRESSION, CHEMICAL; DIMERIZATION; HL-60 CELLS; HUMANS; PYRIMIDINES; RECEPTORS, RETINOIC ACID; RETINOID X RECEPTORS; STRUCTURE-ACTIVITY RELATIONSHIP; TETRAHYDRONAPHTHALENES; TRANSCRIPTION FACTORS;

EID: 0036682057     PISSN: 00222623     EISSN: None     Source Type: Journal    
DOI: 10.1021/jm0255320     Document Type: Article

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