Solid-phase synthesis of unsaturated 3-substituted piperazine-2,5-diones

Journal of Combinatorial Chemistry

Volumn 4, Issue 2, 2002, Pages 106-108

  Li, Wen Ren ^a   Yang, Jian Hsiu ^a  

^a NATIONAL CENTRAL UNIVERSITY   (Taiwan)

Author keywords

[No Author keywords available]

Indexed keywords

ENZYME INHIBITOR; PIPERAZINE DERIVATIVE; PROTEIN TYROSINE KINASE;

ARTICLE; COMBINATORIAL CHEMISTRY; DRUG ANTAGONISM; DRUG STABILITY; SYNTHESIS;

COMBINATORIAL CHEMISTRY TECHNIQUES; DRUG STABILITY; ENZYME INHIBITORS; PIPERAZINES; PROTEIN-TYROSINE KINASES;

EID: 0036512408     PISSN: 15204766     EISSN: None     Source Type: Journal    
DOI: 10.1021/cc010055c     Document Type: Article

References (38)

1. Gallop, M. A.; Barrett, R. W.; Dower, W. J.; Fodor, S. P. A.; Gordon, E. M. J. Med. Chem. 1994, 37, 1233.
2. Gordon, E. M.; Barrett, R. W.; Dower, W. J.; Fodor, S. P. A.; Gallop, M. A. J. Med. Chem. 1994, 37, 1385.
3. Gordon, D. W.; Steele, J. Bioorg. Med. Chem. Lett. 1995, 5, 47.
4. Terrett, N. K.; Gardner, M.; Gordon, D. W.; Kobylecki, R. J.; Steele, J. Tetrahedron 1995, 51, 8135.
5. Thompson, L. A.; Ellman, J. A. Chem. Rev. 1996, 96, 555 and references therein.
6. Balkenhohl, F.; von dem Bussche-Hünnefeld, C.; Lansky, A.; Zechel, C. Angew. Chem., Int. Ed. Engl. 1996, 35, 2288 and references therein.
7. Fruchtel, J. S.; Jung, G. Angew. Chem., Int. Ed. Engl. 1996, 35, 17.
8. Booth, S.; Hermkens, P. H. H.; Ottenheijm, H. C. J.; Rees, D. C. Tetrahedron 1998, 54, 15385.
9. Dolle, R. E.; Nelson, K. H., Jr. J. Comb. Chem. 1999, 1, 235.
10. Franzén, R. G. J. Comb. Chem. 2000, 2, 195.
11. Cheng, S.; Comer, D. D.; Williams, J. P.; Myers, P. L.; Boger, D. L. J. Am. Chem. Soc. 1996, 118, 2567.
12. Hermkens, P. H. H.; Ottenheijm, H. C. J.; Rees, D. Tetrahedron 1996, 52, 4527.
13. Witiak, D. T.; Wei, Y. In Progress in Drug Research; Jucker, E., Ed.; Birkhäuser Verlag: Basel, Switzerland, 1990; Vol. 35, p 249.
14. Hayashi, Y.; Orikasa, S.; Tanaka, K.; Kanoh, K.; Kiso, Y. J. Org. Chem. 2000, 65, 8402.
15. Chai, C. L. L.; King, A. R. Tetrahedron Lett. 1995, 36, 4295.
16. Baures, P. W.; Ojala, W. H.; Costain, W. J.; Ott, M. C.; Pradhan, A.; Gleason, W. B.; Mishra, R. K.; Johnson, R. L. J. Med. Chem. 1997, 40, 3594.
17. Larsen, T. O.; Frisvad, J. C.; Jensen, S. R. Phytochemistry 1992, 31, 1613.
18. Kanoh, K.; Kohno, S.; Asari, T.; Harada, T.; Katada, J.; Muramatsu, M.; Kawashima, H.; Sekiya, H.; Uno, I. Bioorg. Med. Chem. Lett. 1997, 7, 2847.
19. Tsukamoto, S.; Kato, H.; Hirota, H.; Fusetani, N. Tetrahedron 1995, 51, 6687.
20. Nakatsuka, S.-I.; Miyazaki, H.; Goto, T. Tetrahedron Lett. 1980, 21, 2817.
21. Shin, C.-G. Heterocycles 1983, 20, 1407.
22. Scott, B. O.; Siegmund, A. C.; Marlowe, C. K.; Pei, Y.; Spear, K. L. Mol. Diversity 1995, 1, 125.
23. Kowalski, J.; Lipton, M. A. Tetrahedron Lett. 1996, 37, 5839.
24. Szardenings, A. K.; Burkoth, T. S.; Lu, H. H.; Tien, D. W.; Campbell, D. A. Tetrahedron 1997, 53, 6573.
25. Smith, R. A.; Bobko, M. A.; Lee, W. Bioorg. Med. Chem. Lett. 1998, 8, 2369.
26. Del Fresno, M.; Alsina, J.; Royo, M.; Barany, G.; Albericio, F. Tetrahedron Lett. 1998, 39, 2639.
27. Sabatino, G.; Chelli, M.; Mazzucco, S.; Ginanneschi, M.; Papini, A. M. Tetrahedron Lett. 1999, 40, 809.
28. Bianco, A.; Sonksen, C. P.; Roepstorff, P.; Briand, J. P. J. Org. Chem. 2000, 65, 2179.
29. Bianco, A.; Furrer, J.; Limal, D.; Guichard, G.; Elbayed, K.; Raya, J.; Piotto, M.; Briand, J.-P. J. Comb. Chem. 2000, 2, 681.
30. Szardenings, A. K.; Antonenko, V.; Campbell, D. A.; DeFrancisco, N.; Ida, S.; Shi, L.; Sharkov, N.; Tien, D.; Wang, Y.; Navre, M. J. Med. Chem. 1999, 42, 1348.
31. Li, W.-R.; Peng, S.-Z. Tetrahedron Lett. 1998, 39, 7373.
32. Li, W.-R.; Yo, Y.-C; Lin, Y.-S. Tetrahedron 2000, 56, 8867.
33. Dressman, B. A.; Spangle, L. A.; Kaldor, S. W. Tetrahedron Lett. 1996, 37, 937.
34. Cheung, S. T.; Benoiton, N. L. Can. J. Chem. 1977, 55, 906.
35. Léger, R.; Yen, R.; She, M. W.; Lee, V. J.; Hecker, S. J. Tetrahedron Lett. 1998, 39, 4171.
36. Schmidt, U.; Lieberknecht, A.; Wild, J. Synthesis 1988, 159.
37. Papazisis, K. T.; Geromichalos, G. D.; Dimitriadis, K. A.; Kortsaris, A. H. J. Immunol. Methods. 1997, 208, 151.
38. Liu, F.; Jan, K. Y. Free Radic. Biol. Med. 2000, 28, 55.