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Volumn 64, Issue 1, 2002, Pages 1-15

Homologs of 1,2,5-hexahydro-3-one-1H-1,4-diazepine (DAP) as novel dipeptidomimetics and molecular scaffolds: Efficient preparation of synthons

(3) Han, Yinglin a Mierke, Dale F b Chorev, Michael a,c

a HARVARD MEDICAL SCHOOL (United States)

b BROWN UNIVERSITY (United States)

c BETH ISRAEL DEACONESS MEDICAL CENTER (United States)

Author keywords

Benzodiazepines, side chain to backbone cyclization; Cyclic dipeptide; Dipeptidomimetics for drug design; Molecular scaffold

Indexed keywords

ALKYLATION; ATOMS; CARBON; LIBRARIES; REDUCTION;

SYNTHONS;

SCAFFOLDS;

1,2,5 HEXAHYDRO 3 ONE 1H 1,4 DIAZEPINE; DIAZEPINE DERIVATIVE; DIPEPTIDE; UNCLASSIFIED DRUG;

ALKYLATION; ARTICLE; CHIRALITY; CONFORMATION; CYCLIZATION; SEQUENCE HOMOLOGY; STRUCTURE ACTIVITY RELATION; SYNTHESIS;

AZEPINES; BIOPOLYMERS; DIPEPTIDES; MOLECULAR MIMICRY;

EID: 0036290605 PISSN: 00063525 EISSN: None Source Type: Journal
DOI: 10.1002/bip.10079 Document Type: Article

Times cited : (7)

References (47)

1
- 0000327897
- Ariens, E. J., Ed.; Academic Press: New York
- (1980) Drug Design , vol.10 , pp. 119-143
- Farmer, P.S.¹

2
- 0027102818
- (1992) Eur J Biochem , vol.210 , pp. 911-921
- Gurrath, M.¹ Müller, G.² Kessler, H.³ Aumailley, M.⁴ Timpl, R.⁵

3
- 0030768536
- (1997) Angew Chem Int Ed Engl , vol.36 , pp. 1374-1389
- Haubner, R.¹ Finsinger, D.² Kessler, H.³

4
- 0027318541
- (1993) Tetrahedron , pp. 3547-3558
- Marshall, G.R.¹

5
- 0025997018
- (1991) Angew Chem Int Ed Engl , vol.30 , pp. 1278-1301
- Hirschmann, R.¹

6
- 0001019227
- (1986) Can J Chem , vol.64 , pp. 1514-1520
- Belanger, P.C.¹ Dufresne, C.²

7
- 0026470597
- (1992) J Am Chem Soc , vol.114 , pp. 9217-9218
- Hirschmann, R.¹ Nicolaou, K.C.² Pietranico, S.³ Salvino, J.⁴ Leahy, E.M.⁵ Sprengeler, P.A.⁶ Furst, G.⁷ Smith A.B. III⁸

8
- 0027857964
- (1993) J Am Chem Soc , vol.115 , pp. 12550-12559
- Hirschmann, R.¹ Nicolaou, K.C.² Pietranico, S.³ Leahy, E.M.⁴ Salvino, J.⁵ Arison, B.⁶ Cichy, M.A.⁷ Spoors, P.G.⁸ Shakespheare, W.C.⁹ Sprengeler, P.A.¹⁰ Hamley, P.¹¹ Smith A.B. III¹² Reisine, T.¹³ Raynor, K.¹⁴ Maechker, L.¹⁵ Donaldson, C.¹⁶ Vale, W.¹⁷ Freidinger, R.M.¹⁸ Cascieri, M.A.¹⁹ Strader, C.D.²⁰ more..

9
- 33749666016
- (1994) Angew Chem Int Ed Eng , vol.33 , pp. 687-689
- Graf von Roedern, E.¹ Kessler, H.²

10
- 0347190177
- (1996) J Am Chem Soc , vol.118 , pp. 10156-10167
- Graf von Roedern, E.¹ Lohof, E.² Hessler, G.³ Hoffmann, M.⁴ Kessler, H.⁵

11
- 84982506235
- (1992) J Am Chem Soc , vol.114 , pp. 9699-9701
- Hirschmann, R.¹ Sprengeler, P.A.² Kawasaki, T.³ Leahy, J.W.⁴ Shakespeare, W.C.⁵ Smith A.B. III⁶

12
- 0030970551
- (1997) Bioorg Med Chem Lett , vol.5 , pp. 693-705
- Xue, C.B.¹ Roderick, J.J.² Jackson, S.³ Rafalski, M.⁴ Rockwell, A.L.⁵ Mousa, S.A.⁶ Olson, R.E.⁷ DeGrado, W.F.⁸

14
- 0019972014
- (1982) Nature , vol.298 , pp. 759-760
- Romer, D.¹ Buscher, H.H.² Hill, R.C.³ Maurer, R.⁴ Petcher, T.J.⁵ Zeugner, H.⁶ Benson, W.⁷ Finner, E.⁸ Milkowski, W.⁹ Thies, P.W.¹⁰

15
- 0024529827
- (1989) J Med Chem , vol.32 , pp. 13-16
- Bock, M.G.¹ DiPardo, R.M.² Evans, B.E.³ Rittle, K.E.⁴ Whitter, W.L.⁵ Veber, D.F.⁶ Anderson, P.S.⁷ Freidinger, R.M.⁸

16
- 0023222021
- (1987) J Med Chem , vol.30 , pp. 1229-1239
- Evans, B.E.¹ Rittle, K.E.² Bock, M.G.³ DiPardo, R.M.⁴ Freidinger, R.M.⁵ Whitter, W.L.⁶ Lundell, G.F.⁷ Veber, D.F.⁸

17
- 0027964423
- (1994) J Am Chem Soc , vol.116 , pp. 5077-5083
- McDowell, R.S.¹ Blackburn, B.K.² Gadek, T.R.³ McGee, L.R.⁴ Rawson, T.⁵ Reynolds, M.E.⁶ Robarge, K.D.⁷ Somers, T.C.⁸ Thorsett, E.D.⁹ Tischler, M.¹⁰ Webb R.R. II¹¹ Venuti, M.C.¹²

19
- 0026337736
- (1991) Science , vol.254 , pp. 1799-1802
- Hsu, M.C.¹ Schutt, A.D.² Holly, M.³ Slice, L.W.⁴ Sherman, M.I.⁵ Richman, D.D.⁶ Potash, M.J.⁷ Volsky, D.J.⁸

20
- 0027323459
- (1993) Science , vol.260 , pp. 1937-1942
- James, G.L.¹ Goldstein, J.L.² Brown, M.S.³ Rawson, T.E.⁴ Somers, T.C.⁵ McDowell, R.S.⁶ Crowley, C.W.⁷ Lucas, B.K.⁸ Levinson, A.D.⁹ Marsters, J.C.¹⁰

21
- 17144460557
- (1994) Bioorg Med Chem Lett , vol.2 , pp. 949-957
- Marsters, J.C.¹ McDowell, R.S.² Reynolds, M.E.³ Oare, D.A.⁴ Somers, T.C.⁵ Stanley, M.S.⁶ Rawson, T.E.⁷ Struble, M.E.⁸ Burdick, D.J.⁹ Chan, K.S.¹⁰

22
- 0025014499
- (1990) Nature , vol.343 , pp. 470-474
- Pouwels, R.¹ Andries, K.² Desmyter, J.³ Schols, D.⁴ Kukla, M.J.⁵ Breslin, H.J.⁶ Raeymaeckers, A.⁷ Van Gelder, J.⁸ Woestenborghs, R.⁹ Heykants, J.¹⁰

23
- 0028512485
- (1994) Bioorg Med Chem Lett , vol.2 , pp. 897-908
- Bondinell, W.E.¹ Keenan, R.M.² Miller, W.H.³ Ali, F.E.⁴ Allen, A.C.⁵ DeBrosse, C.W.⁶ Eggleston, D.S.⁷ Erhard, K.F.⁸ Haltiwanger, R.C.⁹ Huffman, W.F.¹⁰

24
- 15844379316
- (1996) J Am Chem Soc , vol.118 , pp. 5156-5157
- Goodman, M.¹ Feng, Y.² Melacini, G.³ Taulane, J.P.⁴

25
- 0024560724
- (1989) Proteins , vol.5 , pp. 13-21
- Mutter, M.¹ Hersperger, R.² Gubemator, K.³ Muller, K.⁴

26
- 0031434205
- (1997) Cell Mol Life Sci , vol.53 , pp. 851-863
- Mutter, M.¹ Tuchscherer, G.²

27
- 0030989391
- (1997) J Org Chem , vol.62 , pp. 2527-2534
- Weitz, I.S.¹ Pellegrini, M.² Mierke, D.F.³ Chorev, M.⁴

28
- 0030901961
- (1997) J Am Chem Soc , vol.119 , pp. 2430-2436
- Pellegrini, M.¹ Weitz, I.S.² Chorev, M.³ Mierke, D.F.⁴

29
- 0036290415
- (2002) Biopolymers , vol.64 , pp. 16-25
- Piserchio, A.¹ Han, Y.² Chorev, M.³ Mierke, D.F.⁴

30
- 2142798911
- (1999) Tetrahedron , vol.426 , pp. 12789-12852
- Hanessian, S.¹ McNaughton-Smith, G.² Lombart, H.-G.³ Lubell, W.D.⁴

31
- 0033592497
- (1999) Org Lett , vol.1 , pp. 1225-1228
- Curran, T.P.¹ Marcaurelle, L.A.² O'Sullivan, K.M.³

32
- 0029007370
- (1995) Int J Pept Protein Res , vol.45 , pp. 540-546
- Esser, F.¹ Carpy, A.² Briem, H.³ Koppen, H.⁴ Pook, K.-H.⁵

33
- 0035903517
- (2001) Angew Chem Int Ed , vol.40 , pp. 3361-3364
- Hoffmann, T.¹ Lanig, H.² Waibel, R.³ Gmeiner, P.⁴

34
- 0025921549
- (1991) Int J Pept Protein Res , vol.37 , pp. 468-475
- Kojima, Y.¹ Ikeda, Y.² Kumata, E.³ Maruo, J.⁴ Okamoto, A.⁵ Hirotsu, K.⁶ Shibata, K.⁷ Ohsuka, A.⁸

35
- 0024553640
- (1989) Int J Pept Protein Res , vol.33 , pp. 110-114
- Yamashita, T.¹ Kojima, Y.² Hirotsu, K.³ Oshuka, A.⁴

36
- 0030936052
- (1997) Org Chem , vol.62 , pp. 1016-1022
- Pohlmann, A.¹ Schanen, V.² Guillaume, D.³ Quirion, J.C.⁴ Husson, H.P.J.⁵

37
- 33646825288
- (1982) J Org Chem , vol.47 , pp. 104-109
- Freidinger, R.M.¹ Perlow, D.S.² Veber, D.F.³

38
- 33845279211
- (1988) J Org Chem , vol.53 , pp. 5607-5616
- Zydowsky, T.M.¹ Dellaria J.F., Jr.² Nellans, H.N.³

39
- 0030032034
- (1996) J Med Chem , vol.39 , pp. 494-502
- Robl, J.A.¹ Cimarusti, M.P.² Simpkins, L.M.³ Brown, B.⁴ Ryono, D.E.⁵ Bird, J.E.⁶ Asaad, M.M.⁷ Schaeffer, T.R.⁸ Trippodo, N.C.⁹

40
- 0001217240
- (1988) J Med Chem , vol.31 , pp. 422-428
- Yanagisawa, H.¹ Ishihara, S.² Ando, A.³ Kanazaki, T.⁴ Miyamoto, S.⁵ Koike, H.⁶ Iijima, Y.⁷ Oizumi, K.⁸ Matsushita, Y.⁹ Hata, T.¹⁰

41
- 0027195926
- (1993) Tetrahedron , pp. 3559-3575
- Tuchscherer, G.¹ Domer, B.² Sila, U.³ Kamber, B.⁴ Mutter, M.⁵

42
- 33845185199
- (1989) J Org Chem , vol.54 , pp. 3164-3173
- Wolf, J.-P.¹ Rapoport, H.²

43
- 0000893663
- (1999) Org Lett , vol.1 , pp. 869-871
- Linder, M.R.¹ Podlech, J.²

44
- 0033583197
- (1999) J Org Chem , vol.64 , pp. 1972-1978
- Han, Y.¹ Chorev, M.²

45
- 0026151057
- (1991) Pept Res , vol.4 , pp. 194-199
- Wade, J.D.¹ Bedford, J.² Sheppard, R.C.³ Tregear, G.W.⁴

46
- 0030039282
- (1996) Chem Pharm Bull , vol.44 , pp. 212-214
- Nishino, N.¹ Arai, T.² Ueno, Y.³ Ohba, M.⁴

47
- 12044258245
- (1993) J Am Chem Soc , vol.115 , pp. 4397-4398
- Carpino, L.A.¹

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