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Volumn 10, Issue 8, 2002, Pages 2535-2542

Piperidino-hydrocarbon compounds as novel non-imidazole histamine H3-receptor antagonists

(7) Meier, Galina a Ligneau, Xavier b Pertz, Heinz H a Ganellin, C Robin c Schwartz, Jean Charles d Schunack, Walter a Stark, Holger e

a FREIE UNIVERSITÄT BERLIN (Germany)

b Laboratoire Bioprojet (France)

c UNIVERSITY COLLEGE LONDON (United Kingdom)

d CENTRE PAUL BROCA (France)

e GOETHE UNIVERSITY (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

3 PHENYLPROPYL 3 PIPERIDINOPROPYL ETHER; BUT 3 YNYLBENZENE; BUTYLLITHIUM N,N,N',N' TETRAMETHYLENE ETHYLENEDIAMINE; CIPROXIFAN; ETHYLENEDIAMINE DERIVATIVE; FUB 427; FUB 637; GT 2227; GT 2331; HISTAMINE H3 RECEPTOR ANTAGONIST; LITHIUM DERIVATIVE; N (4 PHENYLBUT 3 YNYL)PIPERIDINE HYDROGEN OXALATE; N (5 PHENYLHEPT 4 YNYL)PIPERIDINE HYDROGEN OXALATE; N (5 PHENYLPENT 4 YNYL)PIPERIDINE HYDROGEN OXALATE; N (5 PHENYLPENTYL)PIPERIDINE HYDROGEN OXALATE; N (6 PHENYLHEX 3 ENYL)PIPERIDINE HYDROGEN OXALATE; N (7 PHENYLHEPT 3 YNYL)PIPERIDINE; N (7 PHENYLHEPTYL)PIPERIDINE HYDROGEN OXALATE; N (8 PHENYLOCTYL)PIPERIDINE HYDROGEN OXALATE; N (9 PHENYLNONYL)PIPERIDINE HYDROGEN OXALATE; N BUT 3 YNYLPIPERIDINE HYDROGEN OXALATE; N HEX 5 YNYLPIPERIDINE; N OCTYLPIPERIDINE HYDROGEN OXALATE; N PENT 4 YNYLPIPERIDINE; N PENT 4 YNYLPIPERIDINE HYDROGEN OXALATE; PENT 4 YNYLBENZENE; PIPERIDINE DERIVATIVE; THIOPERAMIDE; UNCLASSIFIED DRUG; ANTIHISTAMINIC AGENT; HISTAMINE H3 RECEPTOR;

ALKYLATION; ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; DRUG BIOAVAILABILITY; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; NONHUMAN; PROTON NUCLEAR MAGNETIC RESONANCE; ANIMAL; BIOAVAILABILITY; CHEMISTRY; GUINEA PIG; ILEUM; METABOLISM; MOUSE; ORAL DRUG ADMINISTRATION; STRUCTURE ACTIVITY RELATION; SYNTHESIS;

CAVIA PORCELLUS; SUS SCROFA;

ADMINISTRATION, ORAL; ALKYLATION; ANIMALS; BIOLOGICAL AVAILABILITY; GUINEA PIGS; HISTAMINE ANTAGONISTS; ILEUM; MICE; PIPERIDINES; RECEPTORS, HISTAMINE H3; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0036282715 PISSN: 09680896 EISSN: None Source Type: Journal
DOI: 10.1016/S0968-0896(02)00115-3 Document Type: Article

Times cited : (17)

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