Novel 1, 2, 4-oxadiazoles as potent and selective histamine H3 receptor antagonists

Bioorganic and Medicinal Chemistry Letters

Volumn 6, Issue 7, 1996, Pages 833-838

  Clitherow, J W ^a   Beswick, P ^a   Irving, W J ^a   Scopes, D I C ^a   Barnes, J C ^a   Clapham, J ^a   Brown, J D ^a   Evans, D J ^a   Hayes, A G ^a  

^a GLAXOSMITHKLINE   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

1,2,4 OXADIAZOLE DERIVATIVE; 3 [(4 CHLOROPHENYL)METHYL] 5 [2 (1H IMIDAZOL 4 YL)ETHYL] 1,2,4 OXIDAZOLE; CLOBENPROPIT; GR 175737; HISTAMINE H3 RECEPTOR; HISTAMINE H3 RECEPTOR ANTAGONIST; THIOPERAMIDE; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; BLOOD BRAIN BARRIER; BRAIN CORTEX; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; FLUID INTAKE; GUINEA PIG; HEART ATRIUM; ILEUM; MUSCLE CONTRACTION; NONHUMAN; ORAL DRUG ADMINISTRATION; QUANTITATIVE STRUCTURE ACTIVITY RELATION; RAT; SUBCUTANEOUS DRUG ADMINISTRATION; TACHYCARDIA;

EID: 0029965818     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/0960-894X(96)00122-9     Document Type: Article

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