Mechanisms of GABAA receptor blockade by millimolar concentrations of furosemide in isolated rat Purkinje cells

Neuropharmacology

Volumn 42, Issue 7, 2002, Pages 913-921

  Kolbaev, Sergey N ^a   Sharonova, Irina N ^a   Vorobjev, Vladimir S ^a   Skrebitsky, Vladimir G ^a  

^a BRAIN RESEARCH INSTITUTE   (Russian Federation)

Author keywords

Cerebellum; Furosemide; GABA; Open channel block; Patch clamp

Indexed keywords

4 AMINOBUTYRIC ACID RECEPTOR; 4 AMINOBUTYRIC ACID RECEPTOR BLOCKING AGENT; FUROSEMIDE;

ANIMAL CELL; ARTICLE; CONCENTRATION RESPONSE; CONTROLLED STUDY; DISSOCIATION CONSTANT; DRUG ACTIVITY; DRUG MECHANISM; DRUG PROTEIN BINDING; ELECTRIC POTENTIAL; MEMBRANE DEPOLARIZATION; NONHUMAN; PRIORITY JOURNAL; PURKINJE CELL; RAT;

ANIMALS; CEREBELLUM; EVOKED POTENTIALS; FUROSEMIDE; GABA ANTAGONISTS; GAMMA-AMINOBUTYRIC ACID; MALE; MEMBRANE POTENTIALS; PATCH-CLAMP TECHNIQUES; PURKINJE CELLS; RATS; RATS, WISTAR; RECEPTORS, GABA-A;

EID: 0036278004     PISSN: 00283908     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0028-3908(02)00042-4     Document Type: Article

References (38)

1. Drug blockade of open end-plate channels
2. Voltage-dependent interaction of open-channel blocking molecules with gating of NMDA receptors in rat cortical neurons
3. Trapping of glutamate and glycine during open channel block of rat hippocampal neuron NMDA receptors by 9-aminoacridine
4. Trapping channel block of NMDA-activated responses by amantadine and memantine
5. Dynamics of the actions of tetrahydro-9-aminoacridine and 9-aminoacridine on glutamatergic currents: Concentration-jump studies in cultured rat hippocampal neurons
6. a receptors
7. Loop diuretics
8. Improved patch-clamp techniques for high-resolution current recording from cells and cell-free membrane patches
9. Effects of diuretics on GABA-gated chloride current in frog isolated sensory neurones
10. A receptors in acutely dissociated rat striatal and cerebellar neurons
11. Recent advances in GABA research
12. A receptors α4β2γ2 and α6β2γ2
13. Synaptic currents in cerebellar Purkinje cells
14. A receptors
15. Selective antagonist for the cerebellar granule cell-specific γ-aminobutyric acid type A receptor
16. Blockade of open channels by tetrabutylammonium, 9-aminoacridine and tacrine prevents channels closing and desensitization
17. Action of furosemide on GABA- and glycine currents in rat septal cholinergic neurons in culture
18. A receptor subunit mRNAs in the rat brain. II. Olfactory bulb and cerebellum
19. Use-dependent block of excitatory amino acid currents in cultured neurons by ketamine
20. Actions of ketamine, phencyclidine and MK-801 on NMDA receptor currents in cultured mouse hippocampal neurones
21. A-receptor subtypes really occur in the brain?
22. A receptor determined by electron microscopic image analysis
23. The charge carried by single-channel currents of rat cultured muscle cells in the presence of local anaesthetics
24. Local anaesthetics transiently block currents through single acetylcholine-receptor channels
25. The open channel blocking drug, IEM-1460, reveals functionally distinct alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionate receptors in rat brain neurons
26. A receptors in acutely isolated cerebellar Purkinje cells of the rat
27. A receptor subtypes
28. A receptors
29. Probing of NMDA channels with fast blockers
30. A receptor subtype-selective antagonism by furosemide
31. A receptor subtype
32. Vibrodissociation of sliced mammalian nervous tissue
33. Tetrahydroaminoacridine blocks and prolongs NMDA receptor-mediated responses in a voltage-dependent manner
34. A simple perfusion system for patch-clamp studies
35. A receptors containing the α subunit
36. Ionic blockage of sodium channels in nerve
37. A receptor channel-lining residues probed in cysteine mutants
38. Chloride channels of glycine and GABA receptors with blockers: Monte Carlo minimization and structure-activity relationships