Pharmacological modulation of the diazepam-insensitive recombinant γ- aminobutyric acid(A) receptors α4β2γ2 and α6β2γ2

Molecular Pharmacology

Volumn 50, Issue 5, 1996, Pages 1253-1261

  Knoflach, Frédéric ^a,d   Benke, Dietmar ^a   Wang, Yue ^a,e   Scheurer, Louis ^a   Lüddens, Hartmut ^c   Hamilton, Beverly J ^b   Carter, Donald B ^b   Mohler, Hanns ^a   Benson, Jack A ^a  

^a UNIVERSITY OF ZURICH   (Switzerland)

^b PFIZER INC   (United States)

^c JOHANNES GUTENBERG UNIVERSITY   (Germany)

^d F HOFFMANN LA ROCHE LTD   (Switzerland)

^e TRINITY COLLEGE DUBLIN   (Ireland)

Author keywords

[No Author keywords available]

Indexed keywords

4 AMINOBUTYRIC ACID A RECEPTOR; 4 ETHYL 6,7 DIMETHOXY BETA CARBOLINE 3 CARBOXYLIC ACID METHYL ESTER; BRETAZENIL; DIAZEPAM; FLUMAZENIL; PICROTOXIN; RECEPTOR SUBUNIT;

ANIMAL CELL; ARTICLE; CONFORMATIONAL TRANSITION; DOSE RESPONSE; DRUG RECEPTOR BINDING; NONHUMAN; PRIORITY JOURNAL; PROTEIN CONFORMATION; RAT; RECEPTOR AFFINITY; SYNAPTIC TRANSMISSION;

ANIMALS; AZIDES; BENZODIAZEPINES; BENZODIAZEPINONES; BINDING SITES; CARBOLINES; DIAZEPAM; FUROSEMIDE; GABA AGONISTS; GABA ANTAGONISTS; GABA MODULATORS; GAMMA-AMINOBUTYRIC ACID; IMIDAZOLES; KINETICS; MEMBRANE POTENTIALS; RADIOLIGAND ASSAY; RATS; RECEPTORS, GABA-A; RECOMBINANT PROTEINS; SENSITIVITY AND SPECIFICITY; ZINC;

EID: 0029827577     PISSN: 0026895X     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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