SCOPUS 정보 검색 플랫폼

Drug Metabolism and Disposition

Volumn 30, Issue 1, 2002, Pages 96-99

A pharmacophore for human pregnane X receptor ligands

(2) Ekins, S a Erickson, J A a

a ELI LILLY AND COMPANY (United States)

Author keywords

[No Author keywords available]

Indexed keywords

1,4 BIS(3,5 DICHLORO 2 PYRIDYLOXY)BENZENE; 16ALPHA CYANOPREGNENOLONE; ANDROSTANE DERIVATIVE; BENZENE DERIVATIVE; CLOTRIMAZOLE; DEXAMETHASONE; DEXAMETHASONE 21 TERT BUTYLACETATE; DEXAMETHASONE DERIVATIVE; DRUG METABOLIZING ENZYME; GLYCOPROTEIN P; HORMONE RECEPTOR; HYPERFORIN; KAEMPFEROL; LIGAND; LITHOCHOLIC ACID; MIFEPRISTONE; MULTIDRUG RESISTANCE PROTEIN; NIFEDIPINE; PREGNANE DERIVATIVE; PREGNANE X RECEPTOR; PREGNANE X RECEPTOR LIGAND; PREGNANEDIONE; RIFAMPICIN; SCOPOLETIN; SR 12813; TRABECTEDIN; TROGLITAZONE; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; COMPUTER MODEL; CRYSTAL STRUCTURE; DRUG DETERMINATION; DRUG POTENCY; DRUG TRANSPORT; ENZYME REGULATION; HORMONE RECEPTOR INTERACTION; HUMAN; HYDROPHOBICITY; IC 50; LIGAND BINDING; MINIMUM INHIBITORY CONCENTRATION; MOLECULAR SIZE; MULTIDRUG RESISTANCE; PHARMACOPHORE; PRIORITY JOURNAL; PROTEIN DOMAIN; RECEPTOR DOWN REGULATION; RECEPTOR UPREGULATION; SPATIAL ORIENTATION; STRUCTURE ANALYSIS; TRANSCRIPTION REGULATION; X RAY CRYSTALLOGRAPHY;

BINDING SITES; COMPUTER SIMULATION; CRYSTALLOGRAPHY, X-RAY; LIGANDS; MODELS, MOLECULAR; MOLECULAR CONFORMATION; RECEPTORS, CYTOPLASMIC AND NUCLEAR; RECEPTORS, STEROID;

EID: 0036136534 PISSN: 00909556 EISSN: None Source Type: Journal
DOI: 10.1124/dmd.30.1.96 Document Type: Article

Times cited : (165)

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