Medicinal chemistry and chemical biology of new generation taxane antitumor agents

IUBMB Life

Volumn 53, Issue 4-5, 2002, Pages 269-274

  Ojima, Iwao ^a   Geney, Raphaël ^a   Ungureanu, Ioana Maria ^a   Li, Dansu ^a  

^a STONY BROOK UNIVERSITY   (United States)

Author keywords

Anticancer agent; Immunoconjugate; Multidrug resistance; P glycoprotein; Photoaffinity label; Taxane; Tumor activated prodrug

Indexed keywords

ANTIBODY CONJUGATE; ANTINEOPLASTIC AGENT; CYCLOSPORIN A; DOCETAXEL; GLYCOPROTEIN P; MONOCLONAL ANTIBODY; ORTATAXEL; PACLITAXEL; SB T 11033; SB T 12126 MN901; SB T 1213; SB T 121303; SB T 121304; SB T 12136 KS61; SB T 12136 KS77; SB T 12136 KS78; SB T 12136 MN901; SB T 12162; SBT 11033; SBT 1213; SBT 121303; SBT 121304; SBT 12162; TAXANE DERIVATIVE; UNCLASSIFIED DRUG; VERAPAMIL; BRIDGED COMPOUND; DRUG DERIVATIVE; TAXANE; TAXOID;

ANIMAL MODEL; CANCER; CANCER CELL CULTURE; CANCER CHEMOTHERAPY; CELL STRAIN MCF 7; CLINICAL TRIAL; CONFERENCE PAPER; DRUG BINDING SITE; DRUG BIOAVAILABILITY; DRUG CYTOTOXICITY; HUMAN; HUMAN CELL; MOUSE; MULTIDRUG RESISTANCE; NONHUMAN; PHASE 2 CLINICAL TRIAL; PHOTOAFFINITY LABELING; SCID MOUSE; SQUAMOUS CELL CARCINOMA; ANIMAL; BINDING SITE; CANCER TRANSPLANTATION; CHEMICAL MODEL; CHEMICAL STRUCTURE; CHEMISTRY; PROTEIN TERTIARY STRUCTURE; REVIEW;

ANIMAL; ANTIBODIES, MONOCLONAL; ANTINEOPLASTIC AGENTS; BINDING SITES; BRIDGED COMPOUNDS; CLINICAL TRIALS; DRUG RESISTANCE, MULTIPLE; HUMAN; MICE; MODELS, CHEMICAL; MODELS, MOLECULAR; NEOPLASM TRANSPLANTATION; P-GLYCOPROTEIN; PACLITAXEL; PROTEIN STRUCTURE, TERTIARY; ANIMALS; HUMANS; TAXOIDS;

ANIMALIA; MINK CELL FOCUS-FORMING VIRUS;

EID: 0035991721     PISSN: 15216543     EISSN: None     Source Type: Journal    
DOI: 10.1080/15216540212658     Document Type: Conference Paper

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