Antiplasmodial activity and cytotoxicity of bis-, tris-, and tetraquinolines with linear or cyclic amino linkers

Journal of Medicinal Chemistry

Volumn 44, Issue 11, 2001, Pages 1658-1665

  Girault, S ^a   Grellier, P ^b   Berecibar, A ^a,c   Maes, L ^d   Lemiere P ^a   Mouray, E ^b   Davioud Charvet, E ^a   Sergheraert, C ^a  

^a CNRS   (France)

^b MUSÉUM NATIONAL D'HISTOIRE NATURELLE   (France)

^c PFIZER INC   (United States)

^d Virco BVBA   (Belgium)

Author keywords

[No Author keywords available]

Indexed keywords

BISQUINOLINE DERIVATIVE; QUINOLINE DERIVATIVE; TETRAQUINOLINE DERIVATIVE; TRISQUINOLINE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL CELL; ANTIMALARIAL ACTIVITY; ARTICLE; CONTROLLED STUDY; CYCLIZATION; CYTOTOXICITY; DIMERIZATION; DRUG POTENCY; DRUG STRUCTURE; HUMAN; HUMAN CELL; NONHUMAN; PLASMODIUM FALCIPARUM;

ANIMALS; ANTIMALARIALS; CELLS, CULTURED; CHLOROQUINE; DRUG RESISTANCE; HUMANS; MACROPHAGES, PERITONEAL; MICE; PLASMODIUM FALCIPARUM; QUINOLINES;

EID: 0035942506     PISSN: 00222623     EISSN: None     Source Type: Journal    
DOI: 10.1021/jm001096a     Document Type: Article

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