Synthesis and evaluation of hexahydrochrysene and tetrahydrobenzofluorene ligands for the estrogen receptor

Bioorganic and Medicinal Chemistry Letters

Volumn 11, Issue 10, 2001, Pages 1281-1284

  Tedesco, Rosanna ^a   Youngman, Michael K ^a   Wilson, Scott R ^a   Katzenellenbogen, John A ^a  

^a UNIVERSITY OF ILLINOIS AT URBANA CHAMPAIGN   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CHRYSENE DERIVATIVE; ESTROGEN RECEPTOR ALPHA; ESTROGEN RECEPTOR BETA; FLUORENE DERIVATIVE; HEXAHYDROCHRYSENE; TETRAHYDROBENZOFLUORENE; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; DRUG RECEPTOR BINDING; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; GENETIC TRANSCRIPTION; STRUCTURE ACTIVITY RELATION;

CHRYSENES; ESTROGEN RECEPTOR ALPHA; ESTROGEN RECEPTOR BETA; FLUORENES; HUMANS; LIGANDS; MOLECULAR CONFORMATION; POLYCYCLIC COMPOUNDS; PROTEIN BINDING; RECEPTORS, ESTROGEN; STRUCTURE-ACTIVITY RELATIONSHIP; TRANSCRIPTION, GENETIC; TUMOR CELLS, CULTURED;

EID: 0035927191     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(01)00189-5     Document Type: Article

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