Serotonergic effects and extracellular brain levels of eletriptan, zolmitriptan and sumatriptan in rat brain

European Journal of Pharmacology

Volumn 425, Issue 3, 2001, Pages 203-210

  Johnson, David ^a   Rollema, Hans ^a   Schmidt, Anne ^a   McHarg, Aileen ^b  

^a PFIZER INC   (United States)

^b Candidate Research Group   (United Kingdom)

Author keywords

5 HT (5 hydroxytryptamine, serotonin) release; 5 HT1B 1D receptor; Brain level; Eletriptan; Microdialysis; Sumatriptan; Zolmitriptan

Indexed keywords

ELETRIPTAN; SEROTONIN; SEROTONIN 1A RECEPTOR; SEROTONIN 1B AGONIST; SEROTONIN 1B RECEPTOR; SEROTONIN 1D AGONIST; SEROTONIN 1D RECEPTOR; SUMATRIPTAN; ZOLMITRIPTAN;

ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; BRAIN PERFUSION; CONTROLLED STUDY; DIALYSATE; DRUG BRAIN LEVEL; DRUG EFFECT; DRUG EFFICACY; DRUG POTENCY; DRUG RECEPTOR BINDING; MALE; NONHUMAN; PRIORITY JOURNAL; RAT; SEROTONIN RELEASE;

ANIMALS; BINDING, COMPETITIVE; BRAIN; CATTLE; CEREBRAL CORTEX; DOSE-RESPONSE RELATIONSHIP, DRUG; EXTRACELLULAR SPACE; INDOLES; INJECTIONS, INTRAVENOUS; MEMBRANES; MICRODIALYSIS; OXAZOLIDINONES; PYRIDINES; PYRROLIDINES; RATS; RECEPTORS, SEROTONIN; SEROTONIN; SEROTONIN AGONISTS; SUMATRIPTAN; TIME FACTORS; TRYPTAMINES;

EID: 0035903026     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(01)01151-7     Document Type: Article

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