O-silyl triflate-promoted addition of diethyl phosphite to chiral aldonitrones. A rapid access to complex α-amino phosphonates and their N-hydroxy derivatives

Tetrahedron Letters

Volumn 42, Issue 16, 2001, Pages 3033-3036

  De Risi, Carmela ^a   Dondoni, Alessandro ^a   Perrone, Daniela ^a   Pollini, Gian Piero ^a  

^a UNIVERSITY OF FERRARA   (Italy)

Author keywords

Aminophosphonation; Enzyme inhibitors; Nitrones; Peptide mimetics; Phosphonates; Stereoselective synthesis

Indexed keywords

ALDEHYDE DERIVATIVE; ALDONITRONE DERIVATIVE; ALPHA,BETA DIAMINOPHOSPHONIC ACID DERIVATIVE; BENZYL DERIVATIVE; CARBON; DIETHYL PHOSPHITE; N BENZYL NITRONE DERIVATIVE; N BUTYLOXYCARBONYL ALPHA AMINOALDEHYDE DERIVATIVE; N HYDROXYPHOSPHORAMIDIC ACID DERIVATIVE; NITRONE DERIVATIVE; O SILYLTRIFLATE; PHOSPHITE; PHOSPHONIC ACID DERIVATIVE; PHOSPHORAMIDIC ACID DERIVATIVE; PHOSPHORUS; SILANE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL BOND; CHEMICAL REACTION; CHIRALITY; DRUG STRUCTURE; DRUG SYNTHESIS; REACTION ANALYSIS; STEREOCHEMISTRY;

EID: 0035897223     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(01)00363-X     Document Type: Article

References (34)