[3H]SCH 58261, a selective adenosine A(2A) receptor antagonist, is a useful ligand in autoradiographic studies

Journal of Neurochemistry

Volumn 70, Issue 3, 1998, Pages 1210-1216

  Fredholm, Bertil B ^a   Lindström, Karin ^a   Dionisotti, Silvio ^b   Ongini, Ennio ^b  

^a KAROLINSKA INSTITUTE   (Sweden)

^b San Raffaele Science Park   (Italy)

Author keywords

Adenosine A(2A) receptors; Adenosine A1 receptors; CGS 21680; G proteins; Magnesium; Rat brain autoradiography

Indexed keywords

2 [4 (2 CARBOXYETHYL)PHENETHYLAMINO]ADENOSINE 5' (N ETHYLCARBOXAMIDE); 5 AMINO 2 (2 FURYL) 7 (2 PHENYLETHYL)PYRAZOLO[4,3 E][1,2,4]TRIAZOLO[1,5 C]PYRIMIDINE; ADENOSINE 5' (N ETHYLCARBOXAMIDE); ADENOSINE A1 RECEPTOR; ADENOSINE A2A RECEPTOR; ADENOSINE A2A RECEPTOR ANTAGONIST; ADENOSINE DERIVATIVE; CYCLOHEXYLADENOSINE; GUANOSINE TRIPHOSPHATE; MAGNESIUM ION; TRITIUM; ADENOSINE; ADENOSINE RECEPTOR; ANTIHYPERTENSIVE AGENT; DIAGNOSTIC AGENT; DRUG DERIVATIVE; GUANINE NUCLEOTIDE BINDING PROTEIN; LIGAND; MAGNESIUM; PHENETHYLAMINE DERIVATIVE; PYRIMIDINE DERIVATIVE; TRIAZOLE DERIVATIVE;

ANIMAL TISSUE; ARTICLE; AUTORADIOGRAPHY; BINDING AFFINITY; BRAIN; CONCENTRATION RESPONSE; ISOTOPE LABELING; LIGAND BINDING; MALE; NONHUMAN; PRIORITY JOURNAL; RAT; RECEPTOR BINDING; ANIMAL; BINDING COMPETITION; DRUG ANTAGONISM; DRUG POTENTIATION; METABOLISM; METHODOLOGY; RADIOASSAY; SPRAGUE DAWLEY RAT;

ANIMALIA; TRITIUM;

ADENOSINE; ANIMALS; ANTIHYPERTENSIVE AGENTS; AUTORADIOGRAPHY; BINDING, COMPETITIVE; GTP-BINDING PROTEINS; GUANOSINE TRIPHOSPHATE; LIGANDS; MAGNESIUM; MALE; PHENETHYLAMINES; PYRIMIDINES; RADIOLIGAND ASSAY; RATS; RATS, SPRAGUE-DAWLEY; RECEPTOR, ADENOSINE A2A; RECEPTORS, PURINERGIC P1; TRIAZOLES; TRITIUM;

EID: 0031594757     PISSN: 00223042     EISSN: None     Source Type: Journal    
DOI: 10.1046/j.1471-4159.1998.70031210.x     Document Type: Article

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