Binding of [3H]CB 34, a selective ligand for peripheral benzodiazepine receptors, to rat brain membranes

European Journal of Pharmacology

Volumn 432, Issue 2-3, 2001, Pages 129-134

  Pisu, M Giuseppina ^a   Papi, Giacomo ^a   Porcu, Patrizia ^a   Trapani, Giuseppe ^b   Latrofa, Andrea ^b   Biggio, Giovanni ^a,c   Serra, Mariangela ^a  

^a UNIVERSITY OF CAGLIARI   (Italy)

^b UNIVERSITY OF BARI   (Italy)

^c CNR   (Italy)

Author keywords

Benzodiazepine receptor, peripheral; CB 34; Cerebral cortex, rat; Ligand binding; Radiolabeled

Indexed keywords

6,8 DICHLORO 2 (4 CHLOROPHENYL) N,N DIISOPROPYLIMIDAZO[1,2 A]PYRIDINE 3 CARBOXAMIDE; BENZODIAZEPINE RECEPTOR; DIAZEPAM; FLUNITRAZEPAM; LIGAND; PYRIDINE DERIVATIVE; TRITIUM; 4 AMINOBUTYRIC ACID A RECEPTOR; 4' CHLORODIAZEPAM; 4'-CHLORODIAZEPAM; ANTI ANXIETY AGENTS, BENZODIAZEPINE; ANXIOLYTIC AGENT; BENZODIAZEPINE DERIVATIVE; DELORAZEPAM; DIAGNOSTIC AGENT; DRUG DERIVATIVE; FLUMAZENIL; IMIDAZOLE DERIVATIVE; INDOLEACETIC ACID DERIVATIVE; ISOQUINOLINE DERIVATIVE; MEMBRANE PROTEIN; N SEC BUTYL 1 (2 CHLOROPHENYL) N METHYL 3 ISOQUINOLINECARBOXAMIDE; N,N DI N HEXYL 2 (4 FLUOROPHENYL)INDOLE 3 ACETAMIDE; N,N-DI-N-HEXYL-2-(4-FLUOROPHENYL)INDOLE-3-ACETAMIDE; NORDAZEPAM; RECEPTORS, GABA A;

ANIMAL TISSUE; ARTICLE; BRAIN CORTEX; BRAIN MEMBRANE; BRAIN REGION; CONTROLLED STUDY; DISSOCIATION; DRUG BINDING SITE; DRUG MECHANISM; DRUG RECEPTOR BINDING; FEMALE; HYPOTHALAMUS; LIGAND BINDING; NONHUMAN; PRIORITY JOURNAL; RAT; RECEPTOR AFFINITY; ANIMAL; BINDING COMPETITION; BRAIN; DOSE RESPONSE; DRUG EFFECT; MEMBRANE; METABOLISM; RAT STRAIN;

ANIMAL; ANTI-ANXIETY AGENTS, BENZODIAZEPINE; BENZODIAZEPINONES; BINDING, COMPETITIVE; BRAIN; DOSE-RESPONSE RELATIONSHIP, DRUG; FEMALE; FLUMAZENIL; IMIDAZOLES; INDOLEACETIC ACIDS; ISOQUINOLINES; LIGANDS; MEMBRANE PROTEINS; MEMBRANES; NORDAZEPAM; PYRIDINES; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, GABA-A; TRITIUM;

EID: 0035824255     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(01)01478-9     Document Type: Article

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