Antibiotic activity and characterization of BB-3497, a novel peptide deformylase inhibitor

Antimicrobial Agents and Chemotherapy

Volumn 45, Issue 2, 2001, Pages 563-570

  Clements, J M ^a   Beckett, R P ^a   Brown, A ^a   Catlin, G ^a   Lobell, M ^a   Palan, S ^a   Thomas, W ^a   Whittaker, M ^a   Wood, S ^a   Salama, S ^a   Baker, P J ^a   Rodgers, H F ^a   Barynin, V ^a   Rice, D W ^a   Hunter, M G ^a  

^a British Biotech Pharmaceuticals Ltd   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

ACTINONIN; CYSTEINE; HISTIDINE; N (1 TERT BUTYL 2 DIMETHYLAMINO 2 OXOETHYL) 2 (N FORMYL N HYDROXYAMINOMETHYL)HEXANAMIDE; PEPTIDE DEFORMYLASE INHIBITOR;

ANIMAL EXPERIMENT; ANIMAL MODEL; ANTIBIOTIC RESISTANCE; ANTIMICROBIAL ACTIVITY; ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; CRYSTAL STRUCTURE; DOSE RESPONSE; DRUG BINDING; DRUG BIOAVAILABILITY; DRUG POTENCY; DRUG SCREENING; DRUG SELECTIVITY; ENTEROCOCCUS FAECALIS; ESCHERICHIA COLI; MALE; METHICILLIN RESISTANT STAPHYLOCOCCUS AUREUS; MOUSE; NONHUMAN; PRIORITY JOURNAL;

AMIDOHYDROLASES; AMINOPEPTIDASES; ANIMALS; ANTI-BACTERIAL AGENTS; CRYSTALLOGRAPHY, X-RAY; DRUG RESISTANCE, MICROBIAL; ENZYME INHIBITORS; ESCHERICHIA COLI; HYDROXAMIC ACIDS; MICROBIAL SENSITIVITY TESTS; MUTATION; RATS; REVERSE TRANSCRIPTASE POLYMERASE CHAIN REACTION; TIME FACTORS;

EID: 0035143273     PISSN: 00664804     EISSN: None     Source Type: Journal    
DOI: 10.1128/AAC.45.2.563-570.2001     Document Type: Article

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