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Volumn 9, Issue 6, 2001, Pages 1589-1600

Design, synthesis, and biological evaluation of anti-HIV double-drugsconjugates of HIV protease inhibitors with a reverse transcriptase inhibitor through spontaneously cleavable linkers

(8) Matsumoto, Hikaru a Kimura, Tooru a Hamawaki, Tomonori a Kumagai, Akira a Goto, Toshiyuki b Sano, Kouichi b Hayashi, Yoshio a Kiso, Yoshiaki a

a KYOTO PHARMACEUTICAL UNIVERSITY (Japan)

b OSAKA MEDICAL COLLEGE (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

ANTI HUMAN IMMUNODEFICIENCY VIRUS AGENT; KNI 1039; PRODRUG; PROTEINASE INHIBITOR; RNA DIRECTED DNA POLYMERASE INHIBITOR; UNCLASSIFIED DRUG; ZALCITABINE; ZIDOVUDINE;

ANTIVIRAL ACTIVITY; ARTICLE; CONJUGATE; CONTROLLED STUDY; DRUG DESIGN; DRUG POTENTIATION; DRUG RELEASE; DRUG STABILITY; DRUG SYNTHESIS; HUMAN; HUMAN CELL; HUMAN IMMUNODEFICIENCY VIRUS; HUMAN IMMUNODEFICIENCY VIRUS 1; NONHUMAN;

ANIMALS; ANTI-HIV AGENTS; DRUG DESIGN; DRUG EVALUATION, PRECLINICAL; HIV PROTEASE INHIBITORS; HUMANS; PRODRUGS; REVERSE TRANSCRIPTASE INHIBITORS; STRUCTURE-ACTIVITY RELATIONSHIP; THIAZOLES; TUMOR CELLS, CULTURED; ZIDOVUDINE;

EID: 0034935326 PISSN: 09680896 EISSN: None Source Type: Journal
DOI: 10.1016/S0968-0896(01)00045-1 Document Type: Article

Times cited : (34)

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