메뉴 건너뛰기




Volumn 58, Issue 2, 2001, Pages 91-107

Somatostatin analogs

Author keywords

Conformation studies; Peptidomimetics; Peptoid residues; Somatostatin receptor subtypes; Structure activity relationships

Indexed keywords

1 [3 [N (5 BROMO 2 PYRIDYL) N (3,4 DICHLOROBENZYL)AMINO]PROPYL] 3 [3 (4 IMIDAZOLYL)PROPYL]THIOUREA; ANGIOPEPTIN; ASS 51; ASS 52; ASS 53; BETA LACTAM DERIVATIVE; CYCLO(PROLYLPHENYLALANYL DEXTRO TRYPTOPHYLLYSYLTHREONYLPHENYLALANINE); CYCLO(PROLYLPHENYLALANYL DEXTRO TRYPTOPHYLLYSYLTHREONYLPHENYLALANYL); DEXTRO PHENYLALANYLCYSTEINYLTYROSYL DEXTRO TRYPTOPHYLARGINYLTHREONYLPENICILLAMINYLTHREONINAMIDE 2,7 DISULFIDE; DEXTRO PHENYLALANYLCYSTEINYLTYROSYL DEXTRO TRYPTOPHYLLYSYLVALYLCYSTEINYLTHREONINAMIDE 2,7 DISULFIDE; DEXTRO PHENYLALANYLCYSTEINYLTYROSYL DEXTRO TRYPTOPHYLORNITHYLTHREONYLPENICILLAMINYLTHREONINAMIDE 2,7 DISULFIDE; L 054522; L 083087; L 779976; L 796778; L 797591; L 803087; L 817818; LANTHIONINE OCTREOTIDE; N [3 (AMINOMETHYL)CYCLOHEXYLMETHYL] 3 (1H INDOL 3 YL) 2 [(SPIRO[1H INDENE 1,4' PIPERIDIN] 1' YLCARBONYL)AMINO]PROPIONAMIDE; OCTREOTIDE; OCTREOTIDE AMIDE; PRL 2970; PROLINE DERIVATIVE; PTR 3046; SEGLITIDE; SEROTONIN RECEPTOR; SOMATOSTATIN 14; SOMATOSTATIN 28; SOMATOSTATIN DERIVATIVE; SOMATOSTATIN[8 DEXTRO TRYPTOPHAN]; UNCLASSIFIED DRUG; UNINDEXED DRUG; VAPREOTIDE;

EID: 0034905424     PISSN: 1397002X     EISSN: None     Source Type: Journal    
DOI: 10.1034/j.1399-3011.2001.00873.x     Document Type: Review
Times cited : (89)

References (113)
  • 5
    • 0022500305 scopus 로고
    • Somatostatin in the central nervous system: Physiology and pathological modifications
    • (1986) Prog. Neurobiol , vol.27 , pp. 63-100
    • Epelbaum, J.1
  • 18
    • 0029946788 scopus 로고    scopus 로고
    • The role of somatostatin analogues in the treatment of refractory diarrhoea
    • (1996) Digestion , vol.57 , pp. 107-113
    • Farthing, M.J.1
  • 44
    • 0004448264 scopus 로고
    • Conformation-directed design of cyclic somatostatins containing a βVI-turn mimetic
    • (1995) Lett. Peptide Sci , vol.2 , pp. 182-186
    • Tourwe, D.1
  • 51
    • 0015505502 scopus 로고
    • Conformational equlibria in α- and δ-chymotripsin. Energetics and importance of the salt bridge
    • (1972) J. Mol. Biol , vol.64 , pp. 497-509
    • Fersht, A.R.1
  • 60
    • 0027287377 scopus 로고
    • Cloned somatostatin receptors: Identification of subtype-selective peptides and demonstration of high affinity binding of linear peptides
    • (1993) Mol. Pharmacol , vol.43 , pp. 838-844
    • Raynor, K.1    Murphy, W.2    Coy, D.H.3
  • 69
    • 15644375594 scopus 로고    scopus 로고
    • A backbone cyclic, receptor 5 -selective somatostatin analogue: Synthesis, bioactivity, and nuclear magnetic resonance conformational analysis
    • (1998) J. Med. Chem , vol.41 , pp. 919-929
    • Gilon, C.1    Huenges, M.2    Matha, B.3
  • 99
    • 0017198230 scopus 로고
    • Somatostatin and ACTH are peptides with partial antagonist-like selectivity for opiate receptors
    • (1976) Eur. J. Pharmacol , vol.38 , pp. 211-213
    • Terenius, L.1
  • 105
    • 0023792440 scopus 로고
    • Design and synthesis of somatostatin analogues with topographical properties that lead to highly potent and specific μ-opioid receptor antagonists with greatly reduced binding to somatostatin receptors
    • (1988) J. Med. Chem , vol.319 , pp. 2170-2177
    • Kazmierski, W.1    Wire, W.S.2    Lui, G.K.3
  • 108
    • 0023945508 scopus 로고
    • A new approach to receptor ligand design: Synthesis and conformation of a new class of potent and highly selective μ opioid antagonists utilizing tetrahydroisoquinoline carboxylic acid
    • (1988) Tetrahedron , vol.41 , pp. 697-710
    • Kazmierski, W.M.1    Hruby, V.J.2
  • 111
    • 0033997436 scopus 로고    scopus 로고
    • Opiate aromatic pharmacophore structure-activity relationships in CTAP analogs determined by topographical bias, two-dimension NMR, and biological activity assays
    • (2000) J. Med. Chem , vol.43 , pp. 569-580
    • Bonner, G.G.1    Davis, P.2    Stropova, D.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.