Nf449: A subnanomolar potency antagonist at recombinant rat P2X1 receptors

Naunyn-Schmiedeberg's Archives of Pharmacology

Volumn 364, Issue 3, 2001, Pages 285-290

  Braun, Kirsten ^a   Rettinger, Jürgen ^a   Ganso, Matthias ^a   Kassack, Matthias ^b   Hildebrandt, Caren ^a   Ullmann, Heiko ^b   Nickel, Peter ^b   Schmalzing, Günther ^c   Lambrecht, Günter ^a  

^a GOETHE UNIVERSITY   (Germany)

^b UNIVERSITY OF BONN   (Germany)

^c RWTH AACHEN UNIVERSITY   (Germany)

Author keywords

Guinea pig ileum; HEK 293 cells; NF449; P2 receptor antagonists; P2X receptor; P2Y receptor; Rat vas deferens; Xenopus laevis oocytes

Indexed keywords

4,4',4'',4''' [CARBONYLBIS[IMINO 5,1,3 BENZENETRIYLBIS(CARBONYLIMINO)]]TETRAKISBENZENE 1,3 DISULFONIC ACID; ALPHA 1A ADRENERGIC RECEPTOR; ALPHA,BETA METHYLENEADENOSINE TRIPHOSPHATE; HISTAMINE H1 RECEPTOR; MUSCARINIC M3 RECEPTOR; NF 279; NF 449; PURINE P2X RECEPTOR; PURINE P2Y RECEPTOR; RADIOLIGAND; RECOMBINANT RECEPTOR; SULFONIC ACID DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG SPECIFICITY; EMBRYO CELL; GENE OVEREXPRESSION; GUINEA PIG; HUMAN; HUMAN CELL; ILEUM; NONHUMAN; OOCYTE; RAT; SMOOTH MUSCLE; VAS DEFERENS; XENOPUS LAEVIS;

ANIMALS; BENZENESULFONATES; GUINEA PIGS; ILEUM; MALE; MUSCLE CONTRACTION; MUSCLE, SMOOTH; RATS; RECEPTORS, PURINERGIC P2; SURAMIN; VAS DEFERENS; XENOPUS LAEVIS;

EID: 0034876923     PISSN: 00281298     EISSN: None     Source Type: Journal    
DOI: 10.1007/s002100100463     Document Type: Article

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