Synthesis and characterization of a quinolinonic compound activating ATP-sensitive K+ channels in endocrine and smooth muscle tissues

British Journal of Pharmacology

Volumn 134, Issue 2, 2001, Pages 375-385

  Becker, B ^a   Antoine, M H ^a   Nguyen, Q A ^a   Rigo, B ^b   Cosgrove, K E ^c   Barnes, P D ^c   Dunne, M J ^c   Pirotte, B ^d   Lebrun, P ^a  

^a UNIVERSITÉ LIBRE DE BRUXELLES   (Belgium)

^b Ecole des Hautes Etudes d'Ingenieur   (France)

^c UNIVERSITY OF SHEFFIELD   (United Kingdom)

^d UNIVERSITY OF LIÈGE   (Belgium)

Author keywords

Contractile activity; Insulin secretion; Quinolinone

Indexed keywords

6 CHLORO 2 METHYLQUINOLIN 4(1H) ONE; 6 FLUORO 2 METHYLQUINOLIN 4(1H) ONE; ADENOSINE TRIPHOSPHATASE (POTASSIUM); CALCIUM ION; DIAZOXIDE; GLIBENCLAMIDE; GLUCOSE; HEI 712; HEI 713; POTASSIUM CHANNEL; POTASSIUM CHANNEL BLOCKING AGENT; POTASSIUM ION; QUINOLINE DERIVATIVE; QUINOLINONE DERIVATIVE; RUBIDIUM 86; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL TISSUE; AORTA MEDIA; ARTICLE; CALCIUM CELL LEVEL; CALCIUM TRANSPORT; CONCENTRATION RESPONSE; DRUG POTENCY; DRUG SYNTHESIS; ENDOCRINE CELL; INSULIN RELEASE; MATHEMATICAL ANALYSIS; NONHUMAN; PANCREAS ISLET; PATCH CLAMP; PRIORITY JOURNAL; RAT; SMOOTH MUSCLE; SMOOTH MUSCLE CONTRACTILITY; VASODILATATION;

EID: 0034775981     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0704266     Document Type: Article

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