Novel aromatic residues in transmembrane domains IV and V involved in agonist binding at α(1a)-adrenergic receptors

Journal of Biological Chemistry

Volumn 275, Issue 16, 2000, Pages 11698-11705

  Waugh, David J J ^a   Zhao, Ming Ming ^a   Zuscik, Michael J ^a   Perez, Dianne M ^a  

^a LERNER RESEARCH INSTITUTE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

2 [[2 (2,6 DIMETHOXYPHENOXY)ETHYL]AMINOMETHYL] 1,4 BENZODIOXAN; 3 ISOPROPYLAMINO 1 (7 METHYL 4 INDANYLOXY) 2 BUTANOL; 5 METHYLURAPIDIL; ADRENALIN; ALPHA 1 ADRENERGIC RECEPTOR; ALPHA 1 ADRENERGIC RECEPTOR BLOCKING AGENT; ALPHA 1 ADRENERGIC RECEPTOR STIMULATING AGENT; BUPHENINE; CLONIDINE; ISOPRENALINE; METHOXAMINE; ORCIPRENALINE; OXYMETAZOLINE; PHENTOLAMINE; PHENYLEPHRINE; PRAZOSIN; PROPRANOLOL; SALBUTAMOL; THEOPHYLLINE;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; DRUG RECEPTOR BINDING; DRUG STRUCTURE; GENE MUTATION; NONHUMAN; PRIORITY JOURNAL; RECEPTOR BINDING; SITE DIRECTED MUTAGENESIS;

ADRENERGIC ALPHA-AGONISTS; AMINO ACID SEQUENCE; ANIMALS; CELL MEMBRANE; COS CELLS; CRICETINAE; EPHEDRINE; EPINEPHRINE; INOSITOL PHOSPHATES; MODELS, CHEMICAL; MOLECULAR SEQUENCE DATA; MUTAGENESIS, SITE-DIRECTED; PHENYLALANINE; PROTEIN CONFORMATION; RATS; RECEPTORS, ADRENERGIC, ALPHA-1; SEQUENCE ALIGNMENT; STRUCTURE-ACTIVITY RELATIONSHIP;

ANIMALIA; STAPHYLOCOCCUS PHAGE 187;

EID: 0034697157     PISSN: 00219258     EISSN: None     Source Type: Journal    
DOI: 10.1074/jbc.275.16.11698     Document Type: Article

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