Constitutive activation of a single effector pathway: Evidence for multiple activation states of a G protein-coupled receptor

Molecular Pharmacology

Volumn 49, Issue 1, 1996, Pages 112-122

  Perez, Dianne M ^a   Hwa, John ^a   Gaivin, Robert ^a   Mathur, Manjula ^a   Brown, Frank ^b   Graham, Robert M ^c  

^a LERNER RESEARCH INSTITUTE   (United States)

^b GLAXOSMITHKLINE   (United States)

^c ST VINCENT S HOSPITAL   (Australia)

Author keywords

[No Author keywords available]

Indexed keywords

2 (2,6 DIMETHYLANILINO) 2 IMIDAZOLINE; 2 [2 (4 HYDROXYPHENYL)ETHYLAMINOMETHYL]TETRALONE; 2 [[2 (2,6 DIMETHOXYPHENOXY)ETHYL]AMINOMETHYL] 1,4 BENZODIOXAN; 2 AMINO 8 METHOXY 5 METHYLTHIOTETRALIN; 5 METHYLURAPIDIL; ADRENALIN; ALANINE; ALPHA 1 ADRENERGIC RECEPTOR BLOCKING AGENT; ALPHA 1 ADRENERGIC RECEPTOR STIMULATING AGENT; ALPHA 1B ADRENERGIC RECEPTOR; ARACHIDONIC ACID; CIRAZOLINE; CLONIDINE; CYSTEINE; DOBUTAMINE; GLUTAMIC ACID; GUANINE NUCLEOTIDE BINDING PROTEIN; IMIDAZOLINE DERIVATIVE; INOSITOL 1,4,5 TRISPHOSPHATE; INOSITOL PHOSPHATE; METHOXAMINE; NORADRENALIN; OXYMETAZOLINE; PHENETHYLAMINE DERIVATIVE; PHENYLALANINE; PHENYLEPHRINE; PHOSPHOLIPASE A2; PHOSPHOLIPASE C; PRAZOSIN; SKF 43315; UNCLASSIFIED DRUG; UNINDEXED DRUG;

ANIMAL CELL; ARTICLE; CELL STRAIN COS1; CONTROLLED STUDY; DRUG POTENCY; LIGAND BINDING; NONHUMAN; PHOSPHOINOSITIDE METABOLISM; PRIORITY JOURNAL; RECEPTOR BINDING;

ADRENERGIC ALPHA-ANTAGONISTS; ANIMALS; ARACHIDONIC ACID; BASE SEQUENCE; CELL LINE; DNA PRIMERS; GTP-BINDING PROTEINS; INOSITOL 1,4,5-TRISPHOSPHATE; IODINE RADIOISOTOPES; MOLECULAR SEQUENCE DATA; MUTAGENESIS, SITE-DIRECTED; PHENETHYLAMINES; PRAZOSIN; RADIOLIGAND ASSAY; RECEPTORS, ADRENERGIC, ALPHA-1; SIGNAL TRANSDUCTION; TETRALONES; TRITIUM; VIRULENCE FACTORS, BORDETELLA;

EID: 0030049488     PISSN: 0026895X     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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