Synthesis and antibacterial activity of peptide deformylase inhibitors

Biochemistry

Volumn 39, Issue 15, 2000, Pages 4543-4551

  Huntington, Kristi M ^a   Yi, Tian ^a   Wei, Yaoming ^a   Pei, Dehua ^a  

^a OHIO STATE UNIVERSITY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

4 NITROANILINE; ARYLFORMAMIDASE; ENZYME INHIBITOR; FORMYLMETHIONYLLEUCYLPHENYLALANINE; THIOL DERIVATIVE;

ANTIBACTERIAL ACTIVITY; ARTICLE; BACILLUS SUBTILIS; BACTERICIDAL ACTIVITY; BACTERIOLYSIS; DRUG DESIGN; DRUG POTENCY; DRUG SYNTHESIS; DRUG TARGETING; ENTEROCOCCUS FAECALIS; ESCHERICHIA COLI; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; PEPTIDE SYNTHESIS; PRIORITY JOURNAL; STAPHYLOCOCCUS EPIDERMIDIS;

AMIDOHYDROLASES; AMINOPEPTIDASES; ANTI-BACTERIAL AGENTS; BACILLUS SUBTILIS; BACTERIOLYSIS; BINDING, COMPETITIVE; CELL DIVISION; CHELATING AGENTS; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG DESIGN; DRUG RESISTANCE, MICROBIAL; ENTEROCOCCUS FAECALIS; ENZYME INHIBITORS; ESCHERICHIA COLI; HYDROGEN BONDING; MICROBIAL SENSITIVITY TESTS; PEPTIDES; RECOMBINANT PROTEINS; STAPHYLOCOCCUS EPIDERMIDIS; SULFHYDRYL COMPOUNDS; THERMODYNAMICS;

BACILLUS SUBTILIS; BACTERIA (MICROORGANISMS); ENTEROCOCCUS FAECALIS; ESCHERICHIA COLI; NEGIBACTERIA; POSIBACTERIA; STAPHYLOCOCCUS EPIDERMIDIS;

EID: 0034681924     PISSN: 00062960     EISSN: None     Source Type: Journal    
DOI: 10.1021/bi992452y     Document Type: Article

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