A critical residue for isoform difference in tetrodotoxin affinity is a molecular determinant of the external access path for local anesthetics in the cardiac sodium channel

Proceedings of the National Academy of Sciences of the United States of America

Volumn 97, Issue 5, 2000, Pages 2326-2331

  Sunami, Akihiko ^a   Glaaser, Ian W ^a   Fozzard, Harry A ^a  

^a UNIVERSITY OF CHICAGO   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

LIDOCAINE; LOCAL ANESTHETIC AGENT; SODIUM CHANNEL; TETRODOTOXIN;

ANIMAL TISSUE; ARTICLE; BINDING SITE; CONTROLLED STUDY; DRUG BINDING; HEART; LOCAL ANESTHESIA; MEMBRANE PERMEABILITY; MUTATION; NEUROMUSCULAR BLOCKING; NONHUMAN; PRIORITY JOURNAL; RAT;

ANESTHETICS, LOCAL; ANIMALS; BINDING SITES; LIDOCAINE; MUSCLE, SKELETAL; MUTAGENESIS; MYOCARDIUM; PROTEIN ISOFORMS; RATS; SODIUM CHANNELS; TETRODOTOXIN; XENOPUS;

ANIMALIA;

EID: 0034050454     PISSN: 00278424     EISSN: None     Source Type: Journal    
DOI: 10.1073/pnas.030438797     Document Type: Article

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