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Volumn 25, Issue 2, 2000, Pages 159-164

Sitaxsentan sodium. Endothelin ET(A) antagonist treatment of heart failure treatment of pulmonary hypertension

Author keywords

[No Author keywords available]

Indexed keywords

2 BUTYL 7 [2 (2 CARBOXYPROPYL ) 4 METHOXYPHENYL] 5 (3,4 METHYLENEDIOXYPHENYL)CYCLOPENTENO[1,2 B]PYRIDINE; 27 O 3 [2 (3 CARBOXYACRYLOYLAMINO) 5 HYDROXYPHENYL]ACRYLOYLOXY MYRICERONE; 4 (4 METHOXYPHENYL) 2 (3,4 METHYLENEDIOXYPHENYL) 4 OXO 3 (3,4,5 TRIMETHOXYBENZYL) 2 BUTENOIC ACID; ATRASENTAN; BMS 193884; BOSENTAN; CLAZOSENTAN; DARUSENTAN; ENDOTHELIN A RECEPTOR ANTAGONIST; ENDOTHELIN B RECEPTOR ANTAGONIST; ENRASENTAN; SARAFOTOXIN S6C; SITAXENTAN SODIUM; SITAXSENTAN; TAK 044; TEZOSENTAN; UNCLASSIFIED DRUG;

EID: 0034028141     PISSN: 03778282     EISSN: None     Source Type: Journal    
DOI: 10.1358/dof.2000.025.02.567157     Document Type: Review
Times cited : (6)

References (33)
  • 4
    • 0013543367 scopus 로고
    • The human endothelin family: Three structurally and pharmacologically distinct isopeptides predicted by three separate genes
    • Inoue, A., Yanagisawa, M., Kimura, S., Kasuya, Y., Miyauchi, T., Goto. K., Masaki, T. The human endothelin family: Three structurally and pharmacologically distinct isopeptides predicted by three separate genes. Proc Nail Acad Sci USA 1989, 86: 2863-7.
    • (1989) Proc Nail Acad Sci USA , vol.86 , pp. 2863-2867
    • Inoue, A.1    Yanagisawa, M.2    Kimura, S.3    Kasuya, Y.4    Miyauchi, T.5    Goto, K.6    Masaki, T.7
  • 7
    • 0000184085 scopus 로고    scopus 로고
    • TBC11251, a highly selective endothelin-A receptor antagonist, prevents and reverses acute hypoxia-induced pulmonary hypertension in the rat
    • Abst 601
    • Chen, S.J., Brock, T., Stavros, F., Okun, I., Wu, C., Chan, F., Mong, S., Dixon, R.A.F., Oparil, S., Chen, V.F TBC11251, a highly selective endothelin-A receptor antagonist, prevents and reverses acute hypoxia-induced pulmonary hypertension in the rat. FASEB J 1996, 10(3): Abst 601.
    • (1996) FASEB J , vol.10 , Issue.3
    • Chen, S.J.1    Brock, T.2    Stavros, F.3    Okun, I.4    Wu, C.5    Chan, F.6    Mong, S.7    Dixon, R.A.F.8    Oparil, S.9    Chen, V.F.10
  • 8
    • 0031760395 scopus 로고    scopus 로고
    • Systemic administration of the endothelin-A receptor antagonist TBC 11251 attenuates cerebral vasospasm after experimental subarachnoid hemorrhage: Dose study and review of endothelin-based therapies in the literature on cerebral vasospasm
    • Wanebo, J.E., Arthur, A.S., Louis, H.G., West, K., Kassell, N.R, Lee, K.S., Helm, G.A. Systemic administration of the endothelin-A receptor antagonist TBC 11251 attenuates cerebral vasospasm after experimental subarachnoid hemorrhage: Dose study and review of endothelin-based therapies in the literature on cerebral vasospasm. Neurosurgery 1998, 43:1409-17.
    • (1998) Neurosurgery , vol.43 , pp. 1409-1417
    • Wanebo, J.E.1    Arthur, A.S.2    Louis, H.G.3    West, K.4    Kassell, N.R.5    Lee, K.S.6    Helm, G.A.7
  • 9
    • 0342744529 scopus 로고    scopus 로고
    • Inhibition of monocyte/macrophage homing to atherosclerotic plaque by treatment with endothelin receptor-A antagonist
    • Abst 66
    • Pasceri, V., Wu, H., Brock, T., Yeh, E.T.H., Willerson, J.T. Inhibition of monocyte/macrophage homing to atherosclerotic plaque by treatment with endothelin receptor-A antagonist. Circulation 1999, 100(18, Suppl. 1): Abst 66.
    • (1999) Circulation , vol.100 , Issue.18 SUPPL. 1
    • Pasceri, V.1    Wu, H.2    Brock, T.3    Yeh, E.T.H.4    Willerson, J.T.5
  • 16
    • 0343179109 scopus 로고    scopus 로고
    • Texas Biotechnology Company Communication Nov 3
    • TBC-11251 development status. Texas Biotechnology Company Communication Nov 3, 1999.
    • (1999) TBC-11251 Development Status
  • 18
    • 0029945669 scopus 로고    scopus 로고
    • A selective endothelin receptor antagonists. 1. Discovery of A-127722
    • A selective endothelin receptor antagonists. 1. Discovery of A-127722. J Med Chem 1996, 39: 1039-48.
    • (1996) J Med Chem , vol.39 , pp. 1039-1048
    • Winn, M.1    Von Geldern, T.W.2    Opgenorth, T.J.3
  • 19
    • 0032424117 scopus 로고    scopus 로고
    • Pharmacological profile of T-0201, a highly potent and orally active endothelin receptor antagonist
    • Hoshino, T., Yamauchi, R., Kikkawa, K., Yabana, H., Murata, S. Pharmacological profile of T-0201, a highly potent and orally active endothelin receptor antagonist. J Pharmacol Exp Ther 1998, 286: 643-9.
    • (1998) J Pharmacol Exp Ther , vol.286 , pp. 643-649
    • Hoshino, T.1    Yamauchi, R.2    Kikkawa, K.3    Yabana, H.4    Murata, S.5
  • 21
    • 0030980244 scopus 로고    scopus 로고
    • Endothelin receptor antagonists: Effect of serum albumin on potency and comparison of pharmacological characteristics
    • Wu-Wong, J.R., Dixon, D.B., Chiou, W.J., Opgenorth, T.J. Endothelin receptor antagonists: Effect of serum albumin on potency and comparison of pharmacological characteristics. J Pharmacol Exp Ther 1997, 281: 791-8.
    • (1997) J Pharmacol Exp Ther , vol.281 , pp. 791-798
    • Wu-Wong, J.R.1    Dixon, D.B.2    Chiou, W.J.3    Opgenorth, T.J.4
  • 23
    • 0029551537 scopus 로고
    • Pharmacology of L-754,142, a highly potent, orally active, nonpeptidyl endothelin antagonist
    • Williams, D.L. Jr., Murphy. K.L., Nolan, N.A. et al. Pharmacology of L-754,142, a highly potent, orally active, nonpeptidyl endothelin antagonist. J Pharmacol Exp Ther 1995, 275: 1518-26.
    • (1995) J Pharmacol Exp Ther , vol.275 , pp. 1518-1526
    • Williams D.L., Jr.1    Murphy, K.L.2    Nolan, N.A.3
  • 24
    • 0032437265 scopus 로고    scopus 로고
    • Nonpeptide endothelin receptor antagonists XI. Pharmacological characterization of SB 234551, a high-affinity and selective nonpeptide ETA receptor antagonist
    • Ohlstein, E.H., Nambi, P., Hay, D.W., Gellai, M., Brooks, D.P., Luengo, J., Xiang, J.N., Elliott, J.D. Nonpeptide endothelin receptor antagonists XI. Pharmacological characterization of SB 234551, a high-affinity and selective nonpeptide ETA receptor antagonist. J Pharmacol Exp Ther 1998, 286: 650-6.
    • (1998) J Pharmacol Exp Ther , vol.286 , pp. 650-656
    • Ohlstein, E.H.1    Nambi, P.2    Hay, D.W.3    Gellai, M.4    Brooks, D.P.5    Luengo, J.6    Xiang, J.N.7    Elliott, J.D.8
  • 25
    • 0028093424 scopus 로고
    • SB 209670, a rationally designed potent nonpeptide endothelin receptor antagonist
    • Ohlstein, E.H., Nambi, P., Douglas, S.A. et al. SB 209670, a rationally designed potent nonpeptide endothelin receptor antagonist. Proc Natl Acad Sci USA 1994, 91: 8052-6.
    • (1994) Proc Natl Acad Sci USA , vol.91 , pp. 8052-8056
    • Ohlstein, E.H.1    Nambi, P.2    Douglas, S.A.3
  • 26
    • 0030077787 scopus 로고    scopus 로고
    • Nonpeptide endothelin receptor antagonists. VI: Pharmacological characterization of SB 217242, a potent and highly bioavailable endothelin receptor antagonist
    • Ohlstein, E.H., Nambi, P., Lago, A., Hay, D.W., Beck, G., Fong, K.L., Eddy, E.P., Smith, P., Ellens, H., Elliott, J.D. Nonpeptide endothelin receptor antagonists. VI: Pharmacological characterization of SB 217242, a potent and highly bioavailable endothelin receptor antagonist. J Pharmacol Exp Ther 1996, 276: 609-15.
    • (1996) J Pharmacol Exp Ther , vol.276 , pp. 609-615
    • Ohlstein, E.H.1    Nambi, P.2    Lago, A.3    Hay, D.W.4    Beck, G.5    Fong, K.L.6    Eddy, E.P.7    Smith, P.8    Ellens, H.9    Elliott, J.D.10
  • 28
    • 0001271975 scopus 로고    scopus 로고
    • LU 302872 and its racemate (LU 224332) show balanced endothelin-A/B receptor affinity, high oral activity, and inhibit human prostate tissue contractions
    • Raschack, M., Gock, S., Unger, L., Hahn, A., Amberg, W., Jansen, R., Alken, P., Weber, A., Hergenroder, S. LU 302872 and its racemate (LU 224332) show balanced endothelin-A/B receptor affinity, high oral activity, and inhibit human prostate tissue contractions. J Cardiovasc Pharmacol 1998, 31 (Suppl 1.): S241-4.
    • (1998) J Cardiovasc Pharmacol , vol.31 , Issue.SUPPL. 1
    • Raschack, M.1    Gock, S.2    Unger, L.3    Hahn, A.4    Amberg, W.5    Jansen, R.6    Alken, P.7    Weber, A.8    Hergenroder, S.9
  • 29
    • 0029896933 scopus 로고    scopus 로고
    • Discovery and optimization of a novel class of orally active nonpeptidic endothelin-A receptor antagonists
    • Riechers, H., Albrecht, H.P., Amberg, W. et al. Discovery and optimization of a novel class of orally active nonpeptidic endothelin-A receptor antagonists. J Med Chem 1996, 39: 2123-8.
    • (1996) J Med Chem , vol.39 , pp. 2123-2128
    • Riechers, H.1    Albrecht, H.P.2    Amberg, W.3
  • 30
    • 0031456079 scopus 로고    scopus 로고
    • Ro 61-1790, a new hydrosoluble endothelin antagonist: General pharmacology and effects on experimental cerebral vasospasm
    • Roux, S., Breu, V., Giller, T., Neidhart. W., Ramuz, H., Coassolo, P., Clozel, J.P., Clozel, M. Ro 61-1790, a new hydrosoluble endothelin antagonist: General pharmacology and effects on experimental cerebral vasospasm. J Pharmacol Exp Ther 1997, 283: 1110-8.
    • (1997) J Pharmacol Exp Ther , vol.283 , pp. 1110-1118
    • Roux, S.1    Breu, V.2    Giller, T.3    Neidhart, W.4    Ramuz, H.5    Coassolo, P.6    Clozel, J.P.7    Clozel, M.8
  • 31
    • 0013460675 scopus 로고    scopus 로고
    • A receptor antagonist
    • Abst P-143
    • A receptor antagonist. Jpn J Pharmacol 1997, 73(Suppl. 1): Abst P-143.
    • (1997) Jpn J Pharmacol , vol.73 , Issue.SUPPL. 1
    • Mihara, S.1
  • 32
    • 0030440925 scopus 로고    scopus 로고
    • Receptor binding and antagonist properties of a novel endothelin receptor antagonist, TAK-044 cyclo [D-α-aspartyl-3-[(4-phenylpiperazin-1-yl)carbonytl-L-alanyl-L-α- aspartyl-D-2-(2-thienyl)glycyl-L-leucyl-D-tryptophyljdisodium salt], in human endothelinA and endothelinB receptors
    • Masuda, Y., Sugo, T., Kikuchi, T., Kawata, A., Satoh, M., Fujisawa, Y., Itoh, Y., Wakimasu, M., Ohtaki, T Receptor binding and antagonist properties of a novel endothelin receptor antagonist, TAK-044 [cyclo[D-α-aspartyl-3-[(4-phenylpiperazin-1-yl)carbonytl-L-alanyl-L- α-aspartyl-D-2-(2-thienyl)glycyl-L-leucyl-D-tryptophyljdisodium salt], in human endothelinA and endothelinB receptors. J Pharmacol Exp Ther 1996, 279: 675-85.
    • (1996) J Pharmacol Exp Ther , vol.279 , pp. 675-685
    • Masuda, Y.1    Sugo, T.2    Kikuchi, T.3    Kawata, A.4    Satoh, M.5    Fujisawa, Y.6    Itoh, Y.7    Wakimasu, M.8    Ohtaki, T.9


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.