SCOPUS 정보 검색 플랫폼

Volumn 40, Issue 11, 1997, Pages 1690-1697

Discovery of TBC11251, a potent, long acting, orally active endothelin receptor-A selective antagonist

(10) Wu, Chengde a,b Chan, Ming F a Stavros, Fiona a,b Raju, B a,b Okun, Ilya a Mong, Seymour a Keller, Karin M b Brock, Tommy b Kogan, Timothy P b Dixon, Richard A F b

a ImmunoPharmaceutics Inc (United States)

b TEXAS BIOTECHNOLOGY CORPORATION (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ENDOTHELIN A RECEPTOR; ENDOTHELIN A RECEPTOR ANTAGONIST; SITAXSENTAN; UNCLASSIFIED DRUG;

ARTICLE; DRUG ACTIVITY; DRUG BIOAVAILABILITY; DRUG HALF LIFE; DRUG RECEPTOR BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; ORAL DRUG ADMINISTRATION; PHOSPHOINOSITIDE METABOLISM; STRUCTURE ACTIVITY RELATION;

ADMINISTRATION, ORAL; ANIMALS; BINDING, COMPETITIVE; BIOLOGICAL AVAILABILITY; CELL LINE; COS CELLS; DOGS; ENDOTHELIN-1; HALF-LIFE; HUMANS; ISOXAZOLES; MALE; PHOSPHATIDYLINOSITOLS; RATS; RATS, SPRAGUE-DAWLEY; RECEPTOR, ENDOTHELIN A; RECEPTORS, ENDOTHELIN; STRUCTURE-ACTIVITY RELATIONSHIP; THIOPHENES;

EID: 0030943903 PISSN: 00222623 EISSN: None Source Type: Journal
DOI: 10.1021/jm9700068 Document Type: Article

Times cited : (129)

References (8)

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6
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