Transport of valganciclovir, a ganciclovir prodrug, via peptide transporters PEPT1 and PEPT2

Journal of Pharmaceutical Sciences

Volumn 89, Issue 6, 2000, Pages 781-789

  Sugawara, Mitsuru ^a   Huang, Wei ^a   Fei, You Jun ^a   Leibach, Frederick H ^a   Ganapathy, Vadivel ^a   Ganapathy, Malliga E ^a  

^a MEDICAL COLLEGE OF GEORGIA   (United States)

Author keywords

Bioavailability; Ganciclovir; Intestine; Kidney; Peptide transporter; Prodrug; Valyl ester

Indexed keywords

CARRIER PROTEIN; GANCICLOVIR; GLYCYLSARCOSINE; PEPT 1 TRANSPORTER; PEPT 2 TRANSPORTER; PRODRUG; UNCLASSIFIED DRUG; VALGANCICLOVIR;

ARTICLE; BINDING AFFINITY; COMPETITIVE INHIBITION; CYTOMEGALOVIRUS INFECTION; DRUG BIOAVAILABILITY; DRUG INHIBITION; DRUG PROTEIN BINDING; DRUG TRANSPORT; HUMAN; HUMAN CELL;

EID: 0033812228     PISSN: 00223549     EISSN: None     Source Type: Journal    
DOI: 10.1002/(SICI)1520-6017(200006)89:6<781::AID-JPS10>3.0.CO;2-7     Document Type: Article

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