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Volumn 35, Issue 11, 2000, Pages 1001-1010

Ala scan analogues of HOE 140. Synthesis and biological activities

(12) Quartara, Laura a Ricci, Renzo a Meini, Stefania a Patacchini, Riccardo a Giolitti, Alessandro a Amadesi, Silvia b Rizzi, Caterina b Rizzi, Anna b Varani, Katia b Borea, Pier A b A Maggi, Carlo a Regoli, Domenico b

a Menarini Ricerche SpA (Italy)

b UNIVERSITY OF FERRARA (Italy)

Author keywords

Alanine scan; Bioassays correlation; Bradykinin antagonists; Structure activity studies

Indexed keywords

BRADYKININ ANTAGONIST; BRADYKININ B2 RECEPTOR ANTAGONIST; ICATIBANT;

AMINO ACID SUBSTITUTION; ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; BIOASSAY; CHIRALITY; COMPETITIVE INHIBITION; CORRELATION FUNCTION; DRUG ACTIVITY; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; GUINEA PIG; NONHUMAN; STRUCTURE ACTIVITY RELATION;

EID: 0033694076 PISSN: 02235234 EISSN: None Source Type: Journal
DOI: 10.1016/S0223-5234(00)01182-X Document Type: Article

Times cited : (10)

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