Mutations in the B2 bradykinin receptor reveal a different pattern of contacts for peptidic agonists and peptidic antagonists

Journal of Biological Chemistry

Volumn 271, Issue 45, 1996, Pages 28277-28286

  Jarnagin, Kurt ^a   Bhakta, Sunil ^a   Zuppan, Patty ^a   Yee, Calvin ^a   Ho, Teresa ^a   Phan, Thu ^a   Tahilramani, Ram ^a   Pease, Joe H B ^a   Miller, Aaron ^a   Freedman, Richard ^a  

^a ROCHE BIOSCIENCE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

BRADYKININ B2 RECEPTOR; BETA ADRENERGIC RECEPTOR BLOCKING AGENT; BRADYKININ; BRADYKININ RECEPTOR; DRUG DERIVATIVE; ICATIBANT;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; CARBOXY TERMINAL SEQUENCE; COMPETITIVE INHIBITION; DRUG RECEPTOR BINDING; GENE MUTATION; LIGAND BINDING; MOLECULAR MODEL; NONHUMAN; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; PEPTIDE SYNTHESIS; PRIORITY JOURNAL; RECEPTOR AFFINITY; SITE DIRECTED MUTAGENESIS; AMINO ACID SEQUENCE; ANIMAL; BINDING COMPETITION; BINDING SITE; CHEMICAL STRUCTURE; GENETICS; METABOLISM; MOLECULAR GENETICS; POLYMERASE CHAIN REACTION; RAT;

ADRENERGIC BETA-ANTAGONISTS; AMINO ACID SEQUENCE; ANIMALS; BINDING SITES; BINDING, COMPETITIVE; BRADYKININ; MAGNETIC RESONANCE SPECTROSCOPY; MODELS, MOLECULAR; MOLECULAR SEQUENCE DATA; MUTAGENESIS, SITE-DIRECTED; POLYMERASE CHAIN REACTION; RATS; RECEPTOR, BRADYKININ B2; RECEPTORS, BRADYKININ;

EID: 10344255641     PISSN: 00219258     EISSN: None     Source Type: Journal    
DOI: 10.1074/jbc.271.45.28277     Document Type: Article

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