Structural elements of the γ-aminobutyric acid type A receptor conferring subtype selectivity for benzodiazepine site ligands

Journal of Biological Chemistry

Volumn 274, Issue 19, 1999, Pages 13370-13374

  Renard, Stéphane ^a   Olivier, Anne ^b   Granger, Patrick ^b   Avenet, Patrick ^b   Graham, David ^a   Sevrin, Mireille ^b   George, Pascal ^b   Besnard, François ^a  

^a Synthélabo ^*  (France)

^b CNS Research Department   (France)

Author keywords

[No Author keywords available]

Indexed keywords

3 METHYL 6 (3 TRIFLUOROMETHYLPHENYL) 1,2,4 TRIAZOLO[4,3 B]PYRIDAZINE; 4 AMINOBUTYRIC ACID A RECEPTOR; RECEPTOR SUBUNIT; ZOLPIDEM;

AMINO ACID SEQUENCE; AMINO ACID SUBSTITUTION; ARTICLE; LIGAND BINDING; NONHUMAN; PRIORITY JOURNAL; PROTEIN CONFORMATION; RECEPTOR AFFINITY; SITE DIRECTED MUTAGENESIS; STRUCTURE ANALYSIS;

ALLOSTERIC SITE; AMINO ACID SEQUENCE; ANIMALS; BENZODIAZEPINES; BINDING SITES; LIGANDS; MOLECULAR SEQUENCE DATA; MUTAGENESIS, SITE-DIRECTED; PROTEIN CONFORMATION; PYRIDINES; RATS; RECEPTORS, GABA-A; SEQUENCE HOMOLOGY, AMINO ACID;

EID: 0033531940     PISSN: 00219258     EISSN: None     Source Type: Journal    
DOI: 10.1074/jbc.274.19.13370     Document Type: Article

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