A conformational study of ligands for omega modulatory sites of GABA(A) receptors by NOESY NMR spectroscopy and distance geometry.

Bioorganic and Medicinal Chemistry Letters

Volumn 7, Issue 17, 1997, Pages 2277-2282

  Olivier, Anne ^a,b   Sevrin, Mireille ^b   Durant, François ^a   George, Pascal ^b  

^a UNIVERSITY OF NAMUR   (Belgium)

^b SANOFI   (France)

Author keywords

[No Author keywords available]

Indexed keywords

4 AMINOBUTYRIC ACID A RECEPTOR; 4 AMINOBUTYRIC ACID A RECEPTOR STIMULATING AGENT; BENZODIAZEPINE DERIVATIVE; IMIDAZOPYRIDINE DERIVATIVE; LIGAND; RECEPTOR SUBTYPE; ZOLPIDEM;

ARTICLE; CONFORMATION; DRUG RECEPTOR BINDING; MODULATION; NONHUMAN; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; NUCLEAR OVERHAUSER EFFECT; PROTEIN STRUCTURE; RECEPTOR AFFINITY;

EID: 0030931518     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(97)00404-6     Document Type: Article

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