메뉴 건너뛰기




Volumn 127, Issue 8, 1999, Pages 1860-1866

Comparison of changes in the extracellular concentration of noradrenaline in rat frontal cortex induced by sibutramine or d-amphetamine: Modulation by α2-adrenoceptors

Author keywords

2 adrenoceptors; d amphetamine; Frontal cortex; in vivo microdialysis; Noradrenaline; Sibutramine

Indexed keywords

2 (2 METHOXY 1,4 BENZODIOXAN 2 YL) 2 IMIDAZOLINE; ALPHA 2 ADRENERGIC RECEPTOR; ALPHA 2 ADRENERGIC RECEPTOR BLOCKING AGENT; ANTIDEPRESSANT AGENT; CENTRAL STIMULANT AGENT; DEXAMPHETAMINE; NORADRENALIN; SIBUTRAMINE;

EID: 0032791234     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0702720     Document Type: Article
Times cited : (23)

References (38)
  • 3
    • 0026646270 scopus 로고
    • Effects of desipramine and amphetamine on noradrenergic neurotransmission: Electrophysiological studies in the rat brain
    • Curet, O., DE Montigny, C. & Blier, P. (1992). Effects of desipramine and amphetamine on noradrenergic neurotransmission: electrophysiological studies in the rat brain, Eur. J. Pharmacol., 221, 59-70.
    • (1992) Eur. J. Pharmacol. , vol.221 , pp. 59-70
    • Curet, O.1    De Montigny, C.2    Blier, P.3
  • 4
    • 0023182579 scopus 로고
    • 2-adrenoceptors play a major role in the effects of idazoxan on cortical noradrenaline (as measured by in vivo dialysis) in the rat
    • 2-adrenoceptors play a major role in the effects of idazoxan on cortical noradrenaline (as measured by in vivo dialysis) in the rat. J. Pharmacol. Exp. Ther., 241, 642-649.
    • (1987) J. Pharmacol. Exp. Ther. , vol.241 , pp. 642-649
    • Dennis, T.1    L'Heureux, R.2    Carter, C.3    Scatton, B.4
  • 5
    • 0028067527 scopus 로고
    • Regional extracellular norepinephrine responses to amphetamine and cocaine and effects of clonidine pretreatment
    • Florin, S.M., Kuczenski, R. & Segal, D.S. (1994). Regional extracellular norepinephrine responses to amphetamine and cocaine and effects of clonidine pretreatment. Brain. Res., 654, 53-62.
    • (1994) Brain. Res. , vol.654 , pp. 53-62
    • Florin, S.M.1    Kuczenski, R.2    Segal, D.S.3
  • 6
    • 0030613812 scopus 로고    scopus 로고
    • 2-Adrenergic receptor blockade markedly potentiates duloxetine- and fluoxetine-induced increases in noradrenaline, dopamine, and serotonin levels in the frontal cortex of freely-moving rats
    • 2-Adrenergic receptor blockade markedly potentiates duloxetine-and fluoxetine-induced increases in noradrenaline, dopamine, and serotonin levels in the frontal cortex of freely-moving rats. J. Neurochem., 69, 2616-2619.
    • (1997) J. Neurochem. , vol.69 , pp. 2616-2619
    • Gobert, A.1    Rivet, J.M.2    Cistarelli, C.3    Melon, C.4    Millan, M.J.5
  • 7
    • 0015221319 scopus 로고
    • Effects of amphetamine on single cell activity in a catecholamine nucleus, the locus coeruleus
    • Graham, A.W. & Aghajanian, G.K. (1971). Effects of amphetamine on single cell activity in a catecholamine nucleus, the locus coeruleus. Nature, 234, 100-102.
    • (1971) Nature , vol.234 , pp. 100-102
    • Graham, A.W.1    Aghajanian, G.K.2
  • 8
    • 0030831763 scopus 로고    scopus 로고
    • In vivo criteria to differentiate monoamine uptake inhibitors from releasing drugs: Sibutramine is a reuptake inhibitor
    • Gundlah, C., Martin, K.F., Heal, D.J. & Auerbach, S.B. (1997). In vivo criteria to differentiate monoamine uptake inhibitors from releasing drugs: Sibutramine is a reuptake inhibitor. J. Pharmacol. Exp. Ther., 283, 581-591.
    • (1997) J. Pharmacol. Exp. Ther. , vol.283 , pp. 581-591
    • Gundlah, C.1    Martin, K.F.2    Heal, D.J.3    Auerbach, S.B.4
  • 9
    • 0001612783 scopus 로고
    • Effects in the rat of sibutramine on food intake and the behavioural satiety sequence
    • Halford, J.C.G., Heal, D.J. & Blundell, J.E. (1995). Effects in the rat of sibutramine on food intake and the behavioural satiety sequence. Br. J. Pharmacol., 114, 387P.
    • (1995) Br. J. Pharmacol. , vol.114
    • Halford, J.C.G.1    Heal, D.J.2    Blundell, J.E.3
  • 10
    • 0003131905 scopus 로고    scopus 로고
    • The pharmacology of sibutramine, the first serotonin and noradrenaline reuptake inhibitor to be developed for the treatment of obesity
    • Heal, D.J. & Cheetham, S.C. (1997). The pharmacology of sibutramine, the first serotonin and noradrenaline reuptake inhibitor to be developed for the treatment of obesity. La lettre du pharmacologie, 11, (suppl 10), 3-8.
    • (1997) La Lettre du Pharmacologie , vol.11 , Issue.SUPPL. 10 , pp. 3-8
    • Heal, D.J.1    Cheetham, S.C.2
  • 11
    • 0031820091 scopus 로고    scopus 로고
    • Sibutramine: A novel anti-obesity drug. A review of the pharmacological evidence to differentiate it from d-amphetamine and d-fenfluramine
    • Heal, D.J., Aspley, S., Prow, M.R., Jackson, H.C., Martin, K.F. & Cheetham, S.C. (1998a). Sibutramine: a novel anti-obesity drug. A review of the pharmacological evidence to differentiate it from d-amphetamine and d-fenfluramine. Int. J. Obesity, 22, (Suppl 1), S18-S28.
    • (1998) Int. J. Obesity , vol.22 , Issue.SUPPL. 1
    • Heal, D.J.1    Aspley, S.2    Prow, M.R.3    Jackson, H.C.4    Martin, K.F.5    Cheetham, S.C.6
  • 12
    • 0031689401 scopus 로고    scopus 로고
    • A comparison of the effects on central 5-HT function of sibutramine hydrochloride and other weight-modifying agents
    • Heal, D.J., Cheetham, S.C., Prow, M.R., Martin, K.F. & Buckett, W.R. (1998b). A comparison of the effects on central 5-HT function of sibutramine hydrochloride and other weight-modifying agents. Br. J. Pharmacol., 125, 301-308.
    • (1998) Br. J. Pharmacol. , vol.125 , pp. 301-308
    • Heal, D.J.1    Cheetham, S.C.2    Prow, M.R.3    Martin, K.F.4    Buckett, W.R.5
  • 13
    • 0023485296 scopus 로고
    • The effects of peripheral D-amphetamine, 4-OH amphetamine, and epinephrine on maintained discharge in the locus coeruleus with reference to the modulation of learning and memory by these substances
    • Holdefer, R.N. & Jensen, R.A. (1987). The effects of peripheral D-amphetamine, 4-OH amphetamine, and epinephrine on maintained discharge in the locus coeruleus with reference to the modulation of learning and memory by these substances. Brain Res., 417, 108-117.
    • (1987) Brain Res. , vol.417 , pp. 108-117
    • Holdefer, R.N.1    Jensen, R.A.2
  • 14
    • 0030759773 scopus 로고    scopus 로고
    • Investigation of the mechanisms underlying the hypophagic effects of the 5-HT and noradrenaline reuptake inhibitor, sibutramine, in the rat
    • Jackson, H.C., Bearham, M.C., Hutchins, L.J., Mazurkiewicz, S.E., Needham, A.M. & Heal, D.J. (1997a). Investigation of the mechanisms underlying the hypophagic effects of the 5-HT and noradrenaline reuptake inhibitor, sibutramine, in the rat. Br. J. Pharmacol., 121, 1613-1618.
    • (1997) Br. J. Pharmacol. , vol.121 , pp. 1613-1618
    • Jackson, H.C.1    Bearham, M.C.2    Hutchins, L.J.3    Mazurkiewicz, S.E.4    Needham, A.M.5    Heal, D.J.6
  • 15
    • 0030860731 scopus 로고    scopus 로고
    • Comparison of the effects of sibutramine and other monoamine reuptake inhibitors on food intake in the rat
    • Jackson, N.C., Needham, A.M., Hutchins, L.J., Mazurkiewicz, S.E, & Heal, D.J. (1997b). Comparison of the effects of sibutramine and other monoamine reuptake inhibitors on food intake in the rat. Br. J. Pharmacol., 121, 1758-1762.
    • (1997) Br. J. Pharmacol. , vol.121 , pp. 1758-1762
    • Jackson, N.C.1    Needham, A.M.2    Hutchins, L.J.3    Mazurkiewicz, S.E.4    Heal, D.J.5
  • 17
    • 0026635858 scopus 로고
    • Regional norepinephrine response to amphetamine using dialysis: Comparison with caudate dopamine
    • Kuczenski, R. & Segal, D.S. (1992). Regional norepinephrine response to amphetamine using dialysis: Comparison with caudate dopamine. Synapse, 11, 164-169.
    • (1992) Synapse , vol.11 , pp. 164-169
    • Kuczenski, R.1    Segal, D.S.2
  • 18
    • 0017750402 scopus 로고
    • Sixth gaddum memorial lecture, National Institute for Medical Research, Mill Hill, presynaptic receptors and their role in the regulation of transmitter release
    • Langer, S.Z. (1977). Sixth Gaddum memorial lecture, National Institute for Medical Research, Mill Hill, Presynaptic receptors and their role in the regulation of transmitter release. Br. J. Pharmacol., 60, 481-497.
    • (1977) Br. J. Pharmacol. , vol.60 , pp. 481-497
    • Langer, S.Z.1
  • 19
    • 0025193985 scopus 로고
    • Binding of [3H]idazoxan and of its methoxy derivative [3H]RX821002 in human fat cells: [3H]idazoxan but not [3H]RX821002 labels additional non-alpha2-adrenergic binding sites
    • Langin, D., Paris, H. & Lafontan, M. (1990). Binding of [3H]idazoxan and of its methoxy derivative [3H]RX821002 in human fat cells: [3H]idazoxan but not [3H]RX821002 labels additional non-alpha2-adrenergic binding sites, Mol. Pharmacol., 37, 876-885.
    • (1990) Mol. Pharmacol. , vol.37 , pp. 876-885
    • Langin, D.1    Paris, H.2    Lafontan, M.3
  • 21
    • 0022649583 scopus 로고
    • Measurement of endogenous noradrenaline release in the rat cerebral cortex in vivo by transcortical dialysis: Effects of drugs affecting noradrenergic transmission
    • L'Heureux, R.L., Dennis, T., Curet, O. & Scatton, B. (1986). Measurement of endogenous noradrenaline release in the rat cerebral cortex in vivo by transcortical dialysis: Effects of drugs affecting noradrenergic transmission. J. Neurochem., 46, 1794-1801.
    • (1986) J. Neurochem. , vol.46 , pp. 1794-1801
    • L'Heureux, R.L.1    Dennis, T.2    Curet, O.3    Scatton, B.4
  • 22
    • 0024503310 scopus 로고
    • The contribution of metabolites to the rapid and potent down-regulation of rat cortical β-adrenoceptors by the putative antidepressant sibutramine hydrochloride
    • Luscombe, G.P., Hopcroft, R.H., Thomas, P.C. & Buckett, W.R. (1989). The contribution of metabolites to the rapid and potent down-regulation of rat cortical β-adrenoceptors by the putative antidepressant sibutramine hydrochloride. Neuropharmacology, 28, 129-134.
    • (1989) Neuropharmacology , vol.28 , pp. 129-134
    • Luscombe, G.P.1    Hopcroft, R.H.2    Thomas, P.C.3    Buckett, W.R.4
  • 23
    • 0032101087 scopus 로고    scopus 로고
    • The anxiogenic agents, yohimbine and FG 7142, disrupt the noradrenergic response to novelty
    • Mason, K., Heal, D.J. & Stanford, S.C. (1997). The anxiogenic agents, yohimbine and FG 7142, disrupt the noradrenergic response to novelty. Pharm. Biochem Behav., 60, 321-327.
    • (1997) Pharm. Biochem Behav. , vol.60 , pp. 321-327
    • Mason, K.1    Heal, D.J.2    Stanford, S.C.3
  • 24
    • 0031016238 scopus 로고    scopus 로고
    • Modulation of catecholamine release by alpha2-adrenoceptors and I1-imidazoline receptors in rat brain
    • Meana, J.J., Herrera-Marscihtz, M., Goiny, M. & Silveira, R. (1997). Modulation of catecholamine release by alpha2-adrenoceptors and I1-imidazoline receptors in rat brain. Brain. Res., 744, 216-226.
    • (1997) Brain. Res. , vol.744 , pp. 216-226
    • Meana, J.J.1    Herrera-Marscihtz, M.2    Goiny, M.3    Silveira, R.4
  • 26
    • 0016768855 scopus 로고
    • Structure-activity relations for the acceleration of efflux of noradrenaline from adrenergic nerves in rabbit atria by sympathomimetic amines
    • Paton, D.M. (1975). Structure-activity relations for the acceleration of efflux of noradrenaline from adrenergic nerves in rabbit atria by sympathomimetic amines. Can. J. Physiol. Pharmacol., 53, 822-829.
    • (1975) Can. J. Physiol. Pharmacol. , vol.53 , pp. 822-829
    • Paton, D.M.1
  • 28
    • 0026637542 scopus 로고
    • p-chloroamphetamine induces serotonin release through serotonin transporters
    • Rudnick, G. & Wall, S.C. (1992). p-Chloroamphetamine induces serotonin release through serotonin transporters. Biochemistry, 31, 6710-6718.
    • (1992) Biochemistry , vol.31 , pp. 6710-6718
    • Rudnick, G.1    Wall, S.C.2
  • 29
    • 0021891103 scopus 로고
    • Amphetamine's effects on terminal excitability of noradrenergic locus coeruleus neurones are impulse-dependent at low but not high doses
    • Ryan, L.J., Tepper, J.M., Young, S.J. & Groves, P.M. (1985). Amphetamine's effects on terminal excitability of noradrenergic locus coeruleus neurones are impulse-dependent at low but not high doses. Brain Res., 341, 155-163.
    • (1985) Brain Res. , vol.341 , pp. 155-163
    • Ryan, L.J.1    Tepper, J.M.2    Young, S.J.3    Groves, P.M.4
  • 30
    • 0027260870 scopus 로고
    • Neurochemical mechanism of action of anorectic drugs
    • Samanin, R. & Garattini, S. (1993). Neurochemical mechanism of action of anorectic drugs, Pharmacol. Toxicol., 73, 63-68.
    • (1993) Pharmacol. Toxicol. , vol.73 , pp. 63-68
    • Samanin, R.1    Garattini, S.2
  • 31
    • 0022485129 scopus 로고
    • Extra-cellular overflow of neuroactive amino acids during severe insulin-induced hypoglycemia: In vivo dialysis of the rat hippocampus
    • Sandberg, M., Butcher, S.P. & Hagberg, H. (1986), Extra-cellular overflow of neuroactive amino acids during severe insulin-induced hypoglycemia: in vivo dialysis of the rat hippocampus. J. Neurochem., 47, 178-184.
    • (1986) J. Neurochem. , vol.47 , pp. 178-184
    • Sandberg, M.1    Butcher, S.P.2    Hagberg, H.3
  • 33
    • 0032489483 scopus 로고    scopus 로고
    • Effects of anesthetics on norepinephrine release in the hypothalamus paraventricular nucleus region of awake rats
    • Shimokawa, A., Jin, Q.H., Ishizuka, Y., Kunitaka, T., Takasaki, M. & Kannan, H. (1998). Effects of anesthetics on norepinephrine release in the hypothalamus paraventricular nucleus region of awake rats. Neurosci. Lett., 244, 21-24.
    • (1998) Neurosci. Lett. , vol.244 , pp. 21-24
    • Shimokawa, A.1    Jin, Q.H.2    Ishizuka, Y.3    Kunitaka, T.4    Takasaki, M.5    Kannan, H.6
  • 34
    • 0030942814 scopus 로고    scopus 로고
    • Sibutramine: A review of the pharmacology of a novel antiobesity agent
    • Stock, M.J. (1997). Sibutramine: a review of the pharmacology of a novel antiobesity agent. Int. J. Obes., 21 (Suppl. 1), S25-S29.
    • (1997) Int. J. Obes. , vol.21 , Issue.SUPPL. 1
    • Stock, M.J.1
  • 35
    • 0016593641 scopus 로고
    • Inhibition of both noradrenergic and serotonergic neurons in brain by the alpha-adrenergic agonist clonidine
    • Svensson, T.H., Bunney, B.S. & Aghajanian, G.K. (1975). Inhibition of both noradrenergic and serotonergic neurons in brain by the alpha-adrenergic agonist clonidine. Brain. Res., 92, 291-306.
    • (1975) Brain. Res. , vol.92 , pp. 291-306
    • Svensson, T.H.1    Bunney, B.S.2    Aghajanian, G.K.3
  • 36
    • 0025647857 scopus 로고
    • Amphetamine and other psychostimulants reduce pH gradients in midbrain dopaminergic neurons and chromaffin granules: A mechanism of action
    • Sulzer, D. & Rayport, S. (1990). Amphetamine and other psychostimulants reduce pH gradients in midbrain dopaminergic neurons and chromaffin granules: a mechanism of action. Neuron, 5, 797-808.
    • (1990) Neuron , vol.5 , pp. 797-808
    • Sulzer, D.1    Rayport, S.2
  • 37
    • 0025845029 scopus 로고
    • A microdialysis study of the regulation of endogenous noradrenaline release in the rat hippocampus
    • Thomas, D.N. & Holman, R.B. (1991). A microdialysis study of the regulation of endogenous noradrenaline release in the rat hippocampus. J. Neurochem., 56, 1741-1746.
    • (1991) J. Neurochem. , vol.56 , pp. 1741-1746
    • Thomas, D.N.1    Holman, R.B.2
  • 38
    • 0023472827 scopus 로고
    • Effects of halothane and other chlorinated hydrocarbons on alpha2-adrenoceptors in the mouse cortex
    • Wikberg, J.E.S., Hede, A.R. & Post, C. (1987). Effects of halothane and other chlorinated hydrocarbons on alpha2-adrenoceptors in the mouse cortex. Pharmacol. Toxicol., 61, 271-277.
    • (1987) Pharmacol. Toxicol. , vol.61 , pp. 271-277
    • Wikberg, J.E.S.1    Hede, A.R.2    Post, C.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.