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Volumn 27, Issue 8, 1999, Pages 951-955

Repeated oral rifampicin decreases the jejunal permeability of R/S- verapamil in rats

Author keywords

[No Author keywords available]

Indexed keywords

CYTOCHROME; GLUCOSE; NORVERAPAMIL; RIFAMPICIN; VERAPAMIL;

EID: 0032770435     PISSN: 00909556     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article
Times cited : (31)

References (28)
  • 1
    • 0030002504 scopus 로고    scopus 로고
    • Intestinal drug metabolism and anti-transport processes: A potential paradigm shift in oral drug delivery
    • Benet LZ, Wu CY, Hebert MF and Wacher VJ (1996). Intestinal drug metabolism and anti-transport processes: A potential paradigm shift in oral drug delivery. J Control Release 39:139-143.
    • (1996) J Control Release , vol.39 , pp. 139-143
    • Benet, L.Z.1    Wu, C.Y.2    Hebert, M.F.3    Wacher, V.J.4
  • 2
    • 0031914323 scopus 로고    scopus 로고
    • The antibiotic rifampicin is a nonsteroidal ligand and activator of the human glucocorticoid receptor
    • Calleja C, Pascussi JM, Mani JC, Maurel P and Vilarem MJ (1998) The antibiotic rifampicin is a nonsteroidal ligand and activator of the human glucocorticoid receptor [see comments]. Nat Med 4:92-96.
    • (1998) Nat Med , vol.4 , pp. 92-96
    • Calleja, C.1    Pascussi, J.M.2    Mani, J.C.3    Maurel, P.4    Vilarem, M.J.5
  • 3
    • 0029855969 scopus 로고    scopus 로고
    • Comparison between permeability coefficients in rat and human jejunum
    • Fagerholm U, Johansson M and Lennernäs H (1996) Comparison between permeability coefficients in rat and human jejunum. Pharm Res 13:1336-1342.
    • (1996) Pharm Res , vol.13 , pp. 1336-1342
    • Fagerholm, U.1    Johansson, M.2    Lennernäs, H.3
  • 4
    • 0029786432 scopus 로고    scopus 로고
    • Differential induction of prehepatic and hepatic metabolism of verapamil by rifampin
    • Fromm MF, Busse D, Kroemer HK and Eichelbaum M (1996) Differential induction of prehepatic and hepatic metabolism of verapamil by rifampin. Hepatology 24:796-801.
    • (1996) Hepatology , vol.24 , pp. 796-801
    • Fromm, M.F.1    Busse, D.2    Kroemer, H.K.3    Eichelbaum, M.4
  • 5
    • 0026012803 scopus 로고
    • Effects of verapamil enantiomers and major metabolites on the cytotoxicity of vincristine and daunomycin in human lymphoma cell lines
    • Haussermann K, Benz B, Gekeler V, Schumacher K and Eichelbaum M (1991) Effects of verapamil enantiomers and major metabolites on the cytotoxicity of vincristine and daunomycin in human lymphoma cell lines. Eur J Clin Pharmacol 40:53-59.
    • (1991) Eur J Clin Pharmacol , vol.40 , pp. 53-59
    • Haussermann, K.1    Benz, B.2    Gekeler, V.3    Schumacher, K.4    Eichelbaum, M.5
  • 7
    • 0026778218 scopus 로고
    • Predictability of the in vivo metabolism of verapamil from in vitro data: Contribution of individual metabolic pathways and stereoselective aspects
    • Kroemer HK, Echizen H, Heidemann H and Eichelbaum M (1992) Predictability of the in vivo metabolism of verapamil from in vitro data: Contribution of individual metabolic pathways and stereoselective aspects. J Pharmacol Exp Ther 260:1052-1057.
    • (1992) J Pharmacol Exp Ther , vol.260 , pp. 1052-1057
    • Kroemer, H.K.1    Echizen, H.2    Heidemann, H.3    Eichelbaum, M.4
  • 8
    • 0026795241 scopus 로고
    • Regional jejunal perfusion, a new in vivo approach to study oral drug absorption in man
    • Lennernäs H, Ahrenstedt O, Hallgren R, Knutson L, Ryde M and Paalzow LK (1992) Regional jejunal perfusion, a new in vivo approach to study oral drug absorption in man. Pharm Res 9:1243-1251.
    • (1992) Pharm Res , vol.9 , pp. 1243-1251
    • Lennernäs, H.1    Ahrenstedt, O.2    Hallgren, R.3    Knutson, L.4    Ryde, M.5    Paalzow, L.K.6
  • 9
    • 0023919267 scopus 로고
    • Use of laminar flow and unstirred layer models to predict intestinal absorption in the rat
    • Levitt MD, Kneip JM and Levitt DG (1988) Use of laminar flow and unstirred layer models to predict intestinal absorption in the rat. J Clin Invest 81:1365-1369.
    • (1988) J Clin Invest , vol.81 , pp. 1365-1369
    • Levitt, M.D.1    Kneip, J.M.2    Levitt, D.G.3
  • 12
    • 0029758162 scopus 로고    scopus 로고
    • Inducing properties of rifampicin and rifabutin for selected enzyme activities of the cytochrome P-450 and UDP-glucuronosyltransferase superfamilies in female rat liver
    • Oesch F, Arand M, Benedetti MS, Castelli MG and Dostert P (1996) Inducing properties of rifampicin and rifabutin for selected enzyme activities of the cytochrome P-450 and UDP-glucuronosyltransferase superfamilies in female rat liver. J Antimicrob Chemother 37:1111-1119.
    • (1996) J Antimicrob Chemother , vol.37 , pp. 1111-1119
    • Oesch, F.1    Arand, M.2    Benedetti, M.S.3    Castelli, M.G.4    Dostert, P.5
  • 15
    • 0028840847 scopus 로고
    • Possible involvement of multiple P-glycoprotein-mediated efflux systems in the transport of verapamil and other organic cations across rat intestine
    • Saitoh H and Aungst BJ (1995) Possible involvement of multiple P-glycoprotein-mediated efflux systems in the transport of verapamil and other organic cations across rat intestine. Pharm Res 12:1304-1310.
    • (1995) Pharm Res , vol.12 , pp. 1304-1310
    • Saitoh, H.1    Aungst, B.J.2
  • 16
    • 0032519643 scopus 로고    scopus 로고
    • Modulation of P-glycoprotein expression by cytochrome P450 3A inducers in male and female rat livers
    • Salphati L and Benet LZ (1998) Modulation of P-glycoprotein expression by cytochrome P450 3A inducers in male and female rat livers. Biochem Pharmacol 55:387-395.
    • (1998) Biochem Pharmacol , vol.55 , pp. 387-395
    • Salphati, L.1    Benet, L.Z.2
  • 17
    • 0031780252 scopus 로고    scopus 로고
    • Jejunal absorption and metabolism of R/S-verapamil in humans
    • Sandstrom R, Karlsson A, Knutson L and Lennernas H (1998a) Jejunal absorption and metabolism of R/S-verapamil in humans. Pharm Res 15:856-862.
    • (1998) Pharm Res , vol.15 , pp. 856-862
    • Sandstrom, R.1    Karlsson, A.2    Knutson, L.3    Lennernas, H.4
  • 18
    • 0031870979 scopus 로고    scopus 로고
    • The absence of stereoselective P-glycoprotein mediated transport of R/S-verapamil across the rat jejunum
    • Sandstrom R, Karlsson A and Lennernäs H (1998b) The absence of stereoselective P-glycoprotein mediated transport of R/S-verapamil across the rat jejunum. J Pharm Pharmacol 50:729-735.
    • (1998) J Pharm Pharmacol , vol.50 , pp. 729-735
    • Sandstrom, R.1    Karlsson, A.2    Lennernäs, H.3
  • 19
    • 0032585784 scopus 로고    scopus 로고
    • Enantiomeric separation of verapamil and norverapamil using chiral-AGP as the stationary phase
    • in press
    • Sandstrom R, Lennernäs H, Öhlén K and Karlsson A (1999) Enantiomeric separation of verapamil and norverapamil using chiral-AGP as the stationary phase. J Pharm Biomed Anal. in press.
    • (1999) J Pharm Biomed Anal.
    • Sandstrom, R.1    Lennernäs, H.2    Öhlén, K.3    Karlsson, A.4
  • 20
    • 0030059953 scopus 로고    scopus 로고
    • Modulators and substrates of P-glycoprotein and cytochrome P4503A coordinately up-regulate these proteins in human colon carcinoma cells
    • Schuetz EG, Beck WT and Schuetz JD (1996a) Modulators and substrates of P-glycoprotein and cytochrome P4503A coordinately up-regulate these proteins in human colon carcinoma cells. Mol Pharmacol 49:311-318.
    • (1996) Mol Pharmacol , vol.49 , pp. 311-318
    • Schuetz, E.G.1    Beck, W.T.2    Schuetz, J.D.3
  • 21
    • 0029916534 scopus 로고    scopus 로고
    • P-Glycoprotein: A major determinant of rifampicin-inducible expression of cytochrome P4503A in mice and humans
    • Schuetz EG, Schinkel AH, Relling MV and Schuetz JD (1996b) P-Glycoprotein: A major determinant of rifampicin-inducible expression of cytochrome P4503A in mice and humans. Proc Natl Acad Sci USA 93:4001-4005.
    • (1996) Proc Natl Acad Sci USA , vol.93 , pp. 4001-4005
    • Schuetz, E.G.1    Schinkel, A.H.2    Relling, M.V.3    Schuetz, J.D.4
  • 23
    • 0029028792 scopus 로고
    • Overlapping substrate specificities and tissue distribution of cytochrome P450 3A and P-glycoprotein: Implications for drug delivery and activity in cancer chemotherapy
    • Wacher VJ, Wu CY and Benet LZ (1995) Overlapping substrate specificities and tissue distribution of cytochrome P450 3A and P-glycoprotein: Implications for drug delivery and activity in cancer chemotherapy. Mol Carcinog 13:129-134.
    • (1995) Mol Carcinog , vol.13 , pp. 129-134
    • Wacher, V.J.1    Wu, C.Y.2    Benet, L.Z.3
  • 24
    • 0023588109 scopus 로고
    • Identification of glucocorticoid-inducible cytochromes P-450 in the intestinal mucosa of rats and man
    • Watkins PB, Wrighton SA, Schuetz EG, Molowa DT and Guzelian PS (1987) Identification of glucocorticoid-inducible cytochromes P-450 in the intestinal mucosa of rats and man. J Clin Invest 80:1029-1036.
    • (1987) J Clin Invest , vol.80 , pp. 1029-1036
    • Watkins, P.B.1    Wrighton, S.A.2    Schuetz, E.G.3    Molowa, D.T.4    Guzelian, P.S.5
  • 25
  • 26
    • 0016758480 scopus 로고
    • Induction of drug metabolism in man after rifampicin treatment measured by increased hexobarbital and tolbutamide clearance
    • Zilly W, Breimer DD and Richter E (1975) Induction of drug metabolism in man after rifampicin treatment measured by increased hexobarbital and tolbutamide clearance. Eur J Clin Pharmacol 9:219-227.
    • (1975) Eur J Clin Pharmacol , vol.9 , pp. 219-227
    • Zilly, W.1    Breimer, D.D.2    Richter, E.3
  • 28
    • 0017596185 scopus 로고
    • Stimulation of drug metabolism by rifampicin in patients with cirrhosis or cholestasis measured by increased hexobarbital and tolbutamide clearance
    • Zilly W, Breimer DD and Richter E (1977b) Stimulation of drug metabolism by rifampicin in patients with cirrhosis or cholestasis measured by increased hexobarbital and tolbutamide clearance. Eur J Clin Pharmacol 11:287-293.
    • (1977) Eur J Clin Pharmacol , vol.11 , pp. 287-293
    • Zilly, W.1    Breimer, D.D.2    Richter, E.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.