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Volumn 128, Issue 3, 1999, Pages 751-759

Evidence that histamine homologues discriminate between H3-receptors in guinea-pig cerebral cortex and ileum longitudinal muscle myenteric plexus

Author keywords

3H R methylhistamine; Guinea pig cerebral cortex; Histamine H3 receptors; Longitudinal muscle myenteric plexus

Indexed keywords

ALPHA METHYLHISTAMINE; HISTAMINE; HISTAMINE AGONIST; HISTAMINE DERIVATIVE; HISTAMINE H3 RECEPTOR; IMPENTAMINE; UNCLASSIFIED DRUG; VUF 4701; VUF 4732;

EID: 0032698241     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0702861     Document Type: Article
Times cited : (29)

References (50)
  • 3
    • 0027460624 scopus 로고
    • A single amino acid of the cholecystokinin-B/gastrin receptor determines specificity for non-peptide antagonists
    • BEINBORN, M., LEE, Y-M, MCBRIDE, E.W., QUINN, S.M. & KOPIN, A.S. (1993). A single amino acid of the cholecystokinin-B/gastrin receptor determines specificity for non-peptide antagonists. Nature, 362, 348-350.
    • (1993) Nature , vol.362 , pp. 348-350
    • Beinborn, M.1    Lee, Y.-M.2    Mcbride, E.W.3    Quinn, S.M.4    Kopin, A.S.5
  • 5
    • 0017094162 scopus 로고
    • 3H]-dopamine binding associated with dopamine receptors in calf brain membranes
    • 3H]-dopamine binding associated with dopamine receptors in calf brain membranes. Mol. Pharmacol., 12, 800-812.
    • (1976) Mol. Pharmacol. , vol.12 , pp. 800-812
    • Burt, D.R.1    Creese, I.2    Snyder, S.H.3
  • 8
    • 0028809293 scopus 로고
    • 3 receptors in rat cerebral cortical membranes
    • 3 receptors in rat cerebral cortical membranes. Br. J. Pharmacol., 114, 357-363.
    • (1995) Br. J. Pharmacol. , vol.114 , pp. 357-363
    • Clark, E.A.1    Hill, S.J.2
  • 9
  • 13
    • 0019137579 scopus 로고
    • A ternary complex model explains the agonist-specific binding properties of the adenylate cyclase-coupled β-adrenergic receptor
    • DE LEAN, A., STADEL, J.M. & LEFOKOWITZ, R. (1980). A ternary complex model explains the agonist-specific binding properties of the adenylate cyclase-coupled β-adrenergic receptor. J. Biol. Chem., 255, 7108-7117.
    • (1980) J. Biol. Chem. , vol.255 , pp. 7108-7117
    • De Lean, A.1    Stadel, J.M.2    Lefokowitz, R.3
  • 14
    • 0029007377 scopus 로고
    • 2-Substituted histamines with G-protein-stimulatory activity
    • DETERT, H., HAGELUKEN, A., SEIFERT, R. & SCHUNACK, W. (1995). 2-substituted histamines with G-protein-stimulatory activity. Eur. J. Med. Chem., 30, 271-276.
    • (1995) Eur. J. Med. Chem. , vol.30 , pp. 271-276
    • Detert, H.1    Hageluken, A.2    Seifert, R.3    Schunack, W.4
  • 15
    • 0029889083 scopus 로고    scopus 로고
    • 2-Alkyl-substituted histamines and hydroxyethylimidazoles with G-protein-stimulatory activity
    • DETERT, H., LESCHKE, C., TOGEL, W., SEIFERT, R. & SCHUNACK, W. (1996). 2-alkyl-substituted histamines and hydroxyethylimidazoles with G-protein-stimulatory activity. Eur. J. Med. Chem., 31, 397-405.
    • (1996) Eur. J. Med. Chem. , vol.31 , pp. 397-405
    • Detert, H.1    Leschke, C.2    Togel, W.3    Seifert, R.4    Schunack, W.5
  • 18
    • 0001621225 scopus 로고    scopus 로고
    • 3-receptor radioligand binding assays in guinea-pig cerebral cortex and ileum longitudinal muscle myenteric plexus
    • 430P.
    • 3-receptor radioligand binding assays in guinea-pig cerebral cortex and ileum longitudinal muscle myenteric plexus. Br. J. Pharmacol., 122, 430P.
    • (1997) Br. J. Pharmacol. , vol.122
    • Harper, E.A.1    Shankley, N.P.2    Black, J.W.3
  • 21
    • 0017782452 scopus 로고
    • 1 receptors in intestinal smooth muscle
    • 1 receptors in intestinal smooth muscle. Nature, 270, 361-363.
    • (1977) Nature , vol.270 , pp. 361-363
    • Hill, S.J.1    Young, J.M.2
  • 22
    • 0017100335 scopus 로고
    • The mobile receptor hypothesis and "cooperativity" of hormone binding: Application to insulin
    • JACOBS, S. & CUATRECASAS, P. (1976). The mobile receptor hypothesis and "cooperativity" of hormone binding: Application to insulin. Biochim. Biophys. Acta., 433, 482-495.
    • (1976) Biochim. Biophys. Acta. , vol.433 , pp. 482-495
    • Jacobs, S.1    Cuatrecasas, P.2
  • 24
    • 0018650387 scopus 로고
    • Isomerisation of the muscarinic receptor-antagonist complex
    • JARV, J., HEDLUND, B. & BARTFAI, T. (1979). Isomerisation of the muscarinic receptor-antagonist complex. J. Biol. Chem., 254, 5595-5598.
    • (1979) J. Biol. Chem. , vol.254 , pp. 5595-5598
    • Jarv, J.1    Hedlund, B.2    Bartfai, T.3
  • 25
    • 0018862848 scopus 로고
    • A quantitative analysis of beta-adrenergic receptor interactions: Resolution of high and low affinity states of the receptor by computer modelling of ligand binding data
    • KENT, R.S., DELEAN, A. & LEFKOWITZ, R.J. (1980). A quantitative analysis of beta-adrenergic receptor interactions: Resolution of high and low affinity states of the receptor by computer modelling of ligand binding data. Mol. Pharmacol., 17, 14-23.
    • (1980) Mol. Pharmacol. , vol.17 , pp. 14-23
    • Kent, R.S.1    Delean, A.2    Lefkowitz, R.J.3
  • 27
    • 0003656147 scopus 로고
    • ENZFITTER. A non-linear regression data analysis program for the IBM PC
    • LEATHERBARROW, J. (1987). ENZFITTER. A non-linear regression data analysis program for the IBM PC. Biosoft.
    • (1987) Biosoft
    • Leatherbarrow, J.1
  • 28
    • 0028950255 scopus 로고
    • The two-state model of receptor activation
    • LEFF, P. (1995). The two-state model of receptor activation. Trends Pharmacol. Sci., 16, 89-97.
    • (1995) Trends Pharmacol. Sci. , vol.16 , pp. 89-97
    • Leff, P.1
  • 29
    • 0027297275 scopus 로고
    • Constitutive activity of receptors coupled to guanine nucleotide regulatory proteins
    • LEFKOWITZ, R.J., COTECCHIA, S., SAMAMA, P. & COSTA, T. (1993). Constitutive activity of receptors coupled to guanine nucleotide regulatory proteins. Trends in Pharmacol. Sci., 14, 303-307.
    • (1993) Trends in Pharmacol. Sci. , vol.14 , pp. 303-307
    • Lefkowitz, R.J.1    Cotecchia, S.2    Samama, P.3    Costa, T.4
  • 30
    • 0030874745 scopus 로고    scopus 로고
    • Alkyl-substituted amino acid amides and analogous di and triamines: New non-peptide G protein activators
    • LESCHKE, C., STORM, R., BREITWEG-LEHMANN, E., EXNER, T., NURNBERG, B. & SCHUNACK, W. (1997). Alkyl-substituted amino acid amides and analogous di and triamines: New non-peptide G protein activators. J. Med. Chem., 30, 3130-3139.
    • (1997) J. Med. Chem. , vol.30 , pp. 3130-3139
    • Leschke, C.1    Storm, R.2    Breitweg-Lehmann, E.3    Exner, T.4    Nurnberg, B.5    Schunack, W.6
  • 32
    • 0024520619 scopus 로고
    • A new potent and selective non-peptide gastrin antagonist and brain cholecystokinin receptor (CCK-B) ligand: L-365,260
    • LOTTI, V.L. & CHANG, R.S.L. (1989). A new potent and selective non-peptide gastrin antagonist and brain cholecystokinin receptor (CCK-B) ligand: L-365,260, Eur. J. Pharmacol., 162, 273-280.
    • (1989) Eur. J. Pharmacol. , vol.162 , pp. 273-280
    • Lotti, V.L.1    Chang, R.S.L.2
  • 34
    • 0031832206 scopus 로고    scopus 로고
    • Pharmacological classification of adenosine receptor in the sinoatrial and atrioventricular nodes of the guinea-pig
    • MEESTER, B.J., SHANKLEY, N.P., WELSH, N.J., WOOD, J., MEIJLER, F.L. & BLACK, J.W. (1998). Pharmacological classification of adenosine receptor in the sinoatrial and atrioventricular nodes of the guinea-pig. Br. J. Pharmacol., 124, 685-692.
    • (1998) Br. J. Pharmacol. , vol.124 , pp. 685-692
    • Meester, B.J.1    Shankley, N.P.2    Welsh, N.J.3    Wood, J.4    Meijler, F.L.5    Black, J.W.6
  • 35
    • 0019061918 scopus 로고
    • LIGAND: A versatile computerised approach for characterisation of ligand-binding systems
    • MUNSON, P.J. & RODBARD, D. (1980). LIGAND: a versatile computerised approach for characterisation of ligand-binding systems. Anal. Biochem., 107, 220-239.
    • (1980) Anal. Biochem. , vol.107 , pp. 220-239
    • Munson, P.J.1    Rodbard, D.2
  • 36
    • 0026161478 scopus 로고
    • 3-receptor activation inhibits acetylcholine release from guinea-pig myenteric plexus
    • 3-receptor activation inhibits acetylcholine release from guinea-pig myenteric plexus. Agents & Actions, 33, 167-169.
    • (1991) Agents & Actions , vol.33 , pp. 167-169
    • Poli, E.1    Stark, H.2    Bertaccini, G.3
  • 41
    • 0009470005 scopus 로고
    • Multiple interconvertible affinity states of the δ-opioid agonist receptor complex
    • SPAIN, J.W. & COSCIA, C.J. (1987). Multiple interconvertible affinity states of the δ-opioid agonist receptor complex. Proc. Natl. Acad. Sci. U.S.A., 72, 590-594.
    • (1987) Proc. Natl. Acad. Sci. U.S.A. , vol.72 , pp. 590-594
    • Spain, J.W.1    Coscia, C.J.2
  • 45
    • 0018607313 scopus 로고
    • Fundamental difference between the molecular interactions of agonists and antagonists with the β-adrenergic receptor
    • WEILAND, G.A., MINNEMAN, K.P. & MOLINOFF, P.B. (1979). Fundamental difference between the molecular interactions of agonists and antagonists with the β-adrenergic receptor. Nature, 281, 114-117.
    • (1979) Nature , vol.281 , pp. 114-117
    • Weiland, G.A.1    Minneman, K.P.2    Molinoff, P.B.3
  • 46
    • 0023899387 scopus 로고
    • Multiple agonist-affinity states of opioid receptors: Regulation of binding by guanyl nucleotides in guinea-pig cortical, NG108-15 and 7315c cell membranes
    • WERLING, L.L., PUTTFARCKEN, P.S. & COX, B.M. (1988). Multiple agonist-affinity states of opioid receptors: Regulation of binding by guanyl nucleotides in guinea-pig cortical, NG108-15 and 7315c cell membranes. Mol. Pharmacol., 33, 423-431.
    • (1988) Mol. Pharmacol. , vol.33 , pp. 423-431
    • Werling, L.L.1    Puttfarcken, P.S.2    Cox, B.M.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.