2-Alkyl-substituted histamines and hydroxyethylimidazoles with G-protein-stimulatory activity

European Journal of Medicinal Chemistry

Volumn 31, Issue 5, 1996, Pages 397-405

  Detert, H ^a,b   Leschke, C ^a   Togel W ^a   Seifert, R ^a   Schunack, W ^a  

^a FREIE UNIVERSITÄT BERLIN   (Germany)

^b JOHANNES GUTENBERG UNIVERSITY   (Germany)

Author keywords

2 Substituted hydroxyethylimidazole; G protein; GTPase; Histamine H1 receptor

Indexed keywords

2 OCTYLHISTAMINE; 3 (2 HYDROXYETHYL)IMIDAZOLE DERIVATIVE; GUANINE NUCLEOTIDE BINDING PROTEIN; GUANOSINE TRIPHOSPHATASE; HISTAMINE DERIVATIVE; HISTAMINE H2 RECEPTOR; PERTUSSIS TOXIN; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; CELL MEMBRANE; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; ENZYME ACTIVATION; GUINEA PIG; HUMAN; HUMAN CELL; ILEUM; LEUKEMIA CELL LINE; LIPOPHILICITY; NONHUMAN; STRUCTURE ACTIVITY RELATION;

EID: 0029889083     PISSN: 02235234     EISSN: None     Source Type: Journal    
DOI: 10.1016/0223-5234(96)89166-5     Document Type: Article

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