[3H]t-butylbicycloorthobenzoate binding to recombinant α1β2γ(2s) GABA(A) receptor

European Journal of Pharmacology

Volumn 360, Issue 1, 1998, Pages 99-104

  Peričić, Danka ^a   Mirković, Kety ^a   Jazvinšćak, Maja ^a   Besnard, François ^b  

^a RUDER BO KOVI INSTITUTE   (Croatia)

^b SANOFI   (France)

Author keywords

3H TBOB (t 3H butylbicycloorthobenzoate) binding; Dehydroepiandrosterone sulfate; GABA ( aminobutyric acid); GABA(A) receptor, recombinant; Picrotoxin; Thiopental

Indexed keywords

4 AMINOBUTYRIC ACID; 4 AMINOBUTYRIC ACID A RECEPTOR; CONVULSANT AGENT; PICROTOXIN; PRASTERONE SULFATE; RECEPTOR SUBTYPE; RECOMBINANT RECEPTOR; TERT BUTYLBICYCLOORTHOBENZOATE; THIOPENTAL; 4 AMINOBUTYRIC ACID RECEPTOR BLOCKING AGENT; BENZODIAZEPINE RECEPTOR AFFECTING AGENT; DIAGNOSTIC AGENT; FUSED HETEROCYCLIC RINGS; RECOMBINANT PROTEIN; TERT BUTYLBICYCLO 2 BENZOATE; TERT-BUTYLBICYCLO-2-BENZOATE; TRITIUM;

ARTICLE; BINDING SITE; CELL MEMBRANE; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG RECEPTOR BINDING; EMBRYO; GENETIC TRANSFECTION; HUMAN; HUMAN CELL; PRIORITY JOURNAL; RECEPTOR AFFINITY; SCATCHARD PLOT; BINDING COMPETITION; CELL LINE; CYTOLOGY; DOSE RESPONSE; DRUG EFFECT; KIDNEY; METABOLISM; RADIOASSAY; ULTRASTRUCTURE;

BICYCLO COMPOUNDS, HETEROCYCLIC; BINDING, COMPETITIVE; CELL LINE; CELL MEMBRANE; DEHYDROEPIANDROSTERONE SULFATE; DOSE-RESPONSE RELATIONSHIP, DRUG; GABA ANTAGONISTS; GABA MODULATORS; GAMMA-AMINOBUTYRIC ACID; HUMANS; KIDNEY; PICROTOXIN; RADIOLIGAND ASSAY; RECEPTORS, GABA-A; RECOMBINANT PROTEINS; THIOPENTAL; TRITIUM;

EID: 0032582341     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(98)00661-X     Document Type: Article

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