Felbamate inhibits [3H]t-butylbicycloorthobenzoate (TBOB) binding and enhances Cl- current at the Gammaaminobutyric acidA (GABAA) receptor

Journal of Pharmacology and Experimental Therapeutics

Volumn 277, Issue 3, 1996, Pages 1784-1792

  Kume, Akito ^a   Greenfield Jr , L John ^a   Macdonald, Robert L ^a,b   Albin, Roger L ^a  

^a UNIVERSITY OF MICHIGAN MEDICAL SCHOOL   (United States)

^b UNIVERSITY OF MICHIGAN   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

4 AMINOBUTYRIC ACID A RECEPTOR; ANTICONVULSIVE AGENT; CHLORIDE CHANNEL; FELBAMATE; FUSED HETEROCYCLIC RINGS; PROPANEDIOL DERIVATIVE; TERT BUTYLBICYCLO 2 BENZOATE; TERT-BUTYLBICYCLO-2-BENZOATE; 4 AMINOBUTYRIC ACID; BICUCULLINE METHIODIDE; FLUMAZENIL; NEUROSTEROID; PENTOBARBITAL; PICROTOXIN; TERT BUTYLBICYCLOORTHOBENZOATE; ZINC;

ANIMAL; ARTICLE; AUTORADIOGRAPHY; BINDING COMPETITION; DOSE RESPONSE; DRUG EFFECT; MALE; METABOLISM; MOUSE; RAT; SPRAGUE DAWLEY RAT; ANIMAL TISSUE; BINDING SITE; CHLORIDE CURRENT; CONCENTRATION RESPONSE; DISSOCIATION; DRUG POTENTIATION; DRUG RECEPTOR BINDING; ELECTROPHYSIOLOGY; NONHUMAN; PATCH CLAMP; PRIORITY JOURNAL;

ANIMALS; ANTICONVULSANTS; AUTORADIOGRAPHY; BICYCLO COMPOUNDS, HETEROCYCLIC; BINDING, COMPETITIVE; CHLORIDE CHANNELS; DOSE-RESPONSE RELATIONSHIP, DRUG; MALE; MICE; PROPYLENE GLYCOLS; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, GABA-A;

EID: 0030302507     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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