Interaction of allosteric ligands with GABAA receptors containing one, two, or three different subunits

European Journal of Pharmacology

Volumn 301, Issue 1-3, 1996, Pages 207-214

  Zezula, Jürgen ^a   Slany, Astrid ^a   Sieghart, Werner ^a  

^a MEDICAL UNIVERSITY OF VIENNA   (Austria)

Author keywords

Allosteric binding site; GABAA receptor, recombinant; 35S TBPS ( 35S t butylbicyclophosphorothionate); 3H Flunitrazepam; 3H Muscimol

Indexed keywords

4 AMINOBUTYRIC ACID A RECEPTOR; 4 ISOPROPYL 1 PHOSPHO 2,6,7 TRIOXALICYCLO[2.2.2]OCTANE 1 OXIDE; 4' CHLORODIAZEPAM; ALFAXALONE; CLOMETHIAZOLE; DIAZEPAM; ETAZOLATE; ETOMIDATE; FLUNITRAZEPAM; GABAERGIC RECEPTOR AFFECTING AGENT; MUSCIMOL; PENTOBARBITAL; PROPOFOL; RADIOLIGAND; RECEPTOR SUBUNIT; TERT BUTYLBICYCLOPHOSPHOROTHIOATE; UNCLASSIFIED DRUG;

ALLOSTERISM; ARTICLE; BINDING AFFINITY; BINDING SITE; CONTROLLED STUDY; EMBRYO; GENETIC TRANSFECTION; HUMAN; HUMAN CELL; KIDNEY CELL; PRIORITY JOURNAL; RECEPTOR BINDING;

ALLOSTERIC SITE; BICYCLO COMPOUNDS, HETEROCYCLIC; CELL LINE; CONVULSANTS; FLUNITRAZEPAM; GABA AGONISTS; GABA MODULATORS; HUMANS; KIDNEY; MEMBRANES; MUSCIMOL; RADIOLIGAND ASSAY; RECEPTORS, GABA-A;

EID: 0029891220     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/0014-2999(96)00066-0     Document Type: Article

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