Modulation of GABAA receptor tert-[35S]butylbicyclophosphorothionate binding by antagonists: Relationship to patterns of subunit expression

Journal of Neurochemistry

Volumn 66, Issue 5, 1996, Pages 2179-2187

  Korpi, E R ^a   Seeburg, P H ^b   Luddens H ^b,c  

^a Alko Inc   (Finland)

^b UNIVERSITY OF HEIDELBERG   (Germany)

^c JOHANNES GUTENBERG UNIVERSITY   (Germany)

Author keywords

Bicuculline; Brain regional heterogeneity; GABAA receptor subtypes; SR 95531; Tert 35S Butylbicyclophosphorothionate autoradioqraphy

Indexed keywords

3 AMINO 2 (3 CARBOXYPROPYL) 6 (4 METHOXYPHENYL)PYRIDAZINIUM BROMIDE; 4 AMINOBUTYRIC ACID RECEPTOR; 4 AMINOBUTYRIC ACID RECEPTOR BLOCKING AGENT; BICUCULLINE; FUSED HETEROCYCLIC RINGS; PYRIDAZINE DERIVATIVE; SULFUR; TERT BUTYLBICYCLOPHOSPHOROTHIOATE; TERT-BUTYLBICYCLOPHOSPHOROTHIONATE; RECEPTOR SUBTYPE; RECEPTOR SUBUNIT;

ANIMAL; ARTICLE; AUTORADIOGRAPHY; BRAIN; COMPARATIVE STUDY; DRUG EFFECT; MALE; MEMBRANE; METABOLISM; RAT; WISTAR RAT; ANIMAL TISSUE; DRUG BINDING SITE; DRUG RECEPTOR BINDING; GENE EXPRESSION; LIGAND BINDING; NEUROTRANSMITTER RELEASE; NONHUMAN; PRIORITY JOURNAL; PROTEIN DOMAIN; PROTEIN MODIFICATION; RECEPTOR AFFINITY; STOICHIOMETRY;

ANIMALS; AUTORADIOGRAPHY; BICUCULLINE; BICYCLO COMPOUNDS, HETEROCYCLIC; BRAIN; GABA ANTAGONISTS; MALE; MEMBRANES; PYRIDAZINES; RATS; RATS, WISTAR; RECEPTORS, GABA; SULFUR RADIOISOTOPES;

EID: 0029659001     PISSN: 00223042     EISSN: None     Source Type: Journal    
DOI: 10.1046/j.1471-4159.1996.66052179.x     Document Type: Article

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