Design and synthesis of SH3 domain binding ligands: Modifications of the consensus sequence XPpXP

Bioorganic and Medicinal Chemistry Letters

Volumn 8, Issue 22, 1998, Pages 3137-3142

  Witter, David J ^a   Famiglietti, Sara J ^b   Gambier, John C ^b   Castelhano, Arlindo L ^a  

^a Cadus Pharmaceutical Corporation   (United States)

^b NATIONAL JEWISH MEDICAL AND RESEARCH CENTER   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

LACTAM DERIVATIVE; SPIROLACTAM DERIVATIVE; UNCLASSIFIED DRUG;

AMINO ACID SEQUENCE; ARTICLE; PROTEIN STRUCTURE; PROTEIN SYNTHESIS; SEQUENCE ANALYSIS; SEQUENCE HOMOLOGY;

EID: 0032542077     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(98)00577-0     Document Type: Article

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19. + 988.
20. D ∼ 10 μM.