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Volumn 123, Issue 7, 1998, Pages 1425-1433

Validation of Furchgott's method to determine agonist-dependent A1-adenosine receptor reserve in guinea-pig atrium

Author keywords

A1 adenosine receptor; Adenosine; CCPA; Furchgott's method; R PIA; Receptor reserve

Indexed keywords

2 CHLORO 6 N CYCLOPENTYLADENOSINE; 8 CYCLOPENTYL 3 [3 [[4 (FLUOROSULFONYL)BENZOYL]OXY]PROPYL] 1 PROPYL XANTHINE; ADENOSINE A1 RECEPTOR; PHENYLISOPROPYLADENOSINE; RADIOLIGAND; UNCLASSIFIED DRUG; XANTHINE DERIVATIVE;

EID: 0031937838     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0701747     Document Type: Article
Times cited : (28)

References (29)
  • 1
    • 0025663025 scopus 로고
    • Assessment of relative intrinsic activity of Mu-opioid analgesics in vitro by using β-funaltrexamine
    • ADAMS, J.U., PARONIS, C.A. & HOLTZMAN, S.G. (1990). Assessment of relative intrinsic activity of Mu-opioid analgesics in vitro by using β-funaltrexamine. J. Pharmacol. Exp. Ther., 225, 1027-1032.
    • (1990) J. Pharmacol. Exp. Ther. , vol.225 , pp. 1027-1032
    • Adams, J.U.1    Paronis, C.A.2    Holtzman, S.G.3
  • 2
    • 0024473768 scopus 로고
    • 1 adenosine receptors in atrial and ventricular myocardium from diseased human hearts
    • 1 adenosine receptors in atrial and ventricular myocardium from diseased human hearts. Circ. Res., 65, 1201-1211.
    • (1989) Circ. Res. , vol.65 , pp. 1201-1211
    • Bohm, M.1    Pieske, B.2    Ungerer, M.3    Erdmann, E.4
  • 4
    • 0028115969 scopus 로고
    • Epidural bupivacaine/sufentanil therapy for postoperative pain control in patients tolerant to opioid and unresponsive to epidural bupivacaine/morphine
    • DE LEON-CASASOLA, O.A. & LEMA, M.J. (1994). Epidural bupivacaine/sufentanil therapy for postoperative pain control in patients tolerant to opioid and unresponsive to epidural bupivacaine/morphine. Anesthesiology, 80, 303-309.
    • (1994) Anesthesiology , vol.80 , pp. 303-309
    • De Leon-Casasola, O.A.1    Lema, M.J.2
  • 6
    • 0029040497 scopus 로고
    • The effect of intrinsic efficacy on opioid tolerance
    • DUTTAROY, A. & YOBURN, B.C. (1995). The effect of intrinsic efficacy on opioid tolerance. Anesthesiology, 82, 1226-1236.
    • (1995) Anesthesiology , vol.82 , pp. 1226-1236
    • Duttaroy, A.1    Yoburn, B.C.2
  • 7
    • 0023103968 scopus 로고
    • Coupling of the muscarinic receptors to adenylate cyclase in the rabbit myocardium: Effects of receptor inactivation
    • EHLERT, F.J. (1987). Coupling of the muscarinic receptors to adenylate cyclase in the rabbit myocardium: effects of receptor inactivation. J. Pharmacol. Exp. Ther., 240, 23-30.
    • (1987) J. Pharmacol. Exp. Ther. , vol.240 , pp. 23-30
    • Ehlert, F.J.1
  • 8
    • 0002355204 scopus 로고
    • The use of β-haloalkylamines in the differentiation of receptors and in the determination of dissociation constants of receptor-agonist complexes
    • ed Harper, N.J. & Simmonds, A.B. New York: Academic Press
    • FURCHGOTT, R.F. (1966). The use of β-haloalkylamines in the differentiation of receptors and in the determination of dissociation constants of receptor-agonist complexes. In Advances in Drug Research. Vol. 3, ed Harper, N.J. & Simmonds, A.B. pp. 21-55. New York: Academic Press.
    • (1966) Advances in Drug Research , vol.3 , pp. 21-55
    • Furchgott, R.F.1
  • 9
    • 84981848149 scopus 로고
    • Comparison of dissociation constants and of relative efficacies of selected agonists acting on parasympathetic receptors
    • FURCHGOTT, R.F. & BURSZTYN, P. (1967). Comparison of dissociation constants and of relative efficacies of selected agonists acting on parasympathetic receptors. Ann. New York Acad. Sci., 144, 882-899.
    • (1967) Ann. New York Acad. Sci. , vol.144 , pp. 882-899
    • Furchgott, R.F.1    Bursztyn, P.2
  • 10
    • 0022507177 scopus 로고
    • Receptor reserve in the calcium-dependent cyclic AMP response of astrocytoma cells to muscarinic receptor stimulation: Demonstration by agonist-induced desensitization, receptor inactivation, and phorbol ester treatment
    • HARDEN, T.K., HENG, M. & BROWN, J.H. (1986). Receptor reserve in the calcium-dependent cyclic AMP response of astrocytoma cells to muscarinic receptor stimulation: Demonstration by agonist-induced desensitization, receptor inactivation, and phorbol ester treatment. Mol. Pharmacol., 30, 200-206.
    • (1986) Mol. Pharmacol. , vol.30 , pp. 200-206
    • Harden, T.K.1    Heng, M.2    Brown, J.H.3
  • 11
    • 0020683629 scopus 로고
    • Effects on in vivo β-adrenoceptor down-regulation on cardiac responses to prenalterol and pirbuterol
    • KENAKIN, T.P. & FERRIS, R.M. (1983). Effects on in vivo β-adrenoceptor down-regulation on cardiac responses to prenalterol and pirbuterol. J. Cardiovasc. Pharmacol., 5, 90-97.
    • (1983) J. Cardiovasc. Pharmacol. , vol.5 , pp. 90-97
    • Kenakin, T.P.1    Ferris, R.M.2
  • 13
    • 0021211721 scopus 로고
    • The Classification of drugs and drug receptors in isolated tissues
    • KENAKIN, T.P. (1984). The Classification of drugs and drug receptors in isolated tissues. Pharmacol. Rev., 36, 165-222.
    • (1984) Pharmacol. Rev. , vol.36 , pp. 165-222
    • Kenakin, T.P.1
  • 14
    • 0023009431 scopus 로고
    • 1 adenosine receptors: Persistent activation reveal spare receptors
    • 1 adenosine receptors: persistent activation reveal spare receptors. Mol. Pharmacol., 30, 403-409.
    • (1986) Mol. Pharmacol. , vol.30 , pp. 403-409
    • Lohse, M.J.1    Klotz, K.-N.2    Schwabe, U.3
  • 15
    • 0021895303 scopus 로고
    • Demonstration of Ri-type adenosine receptors in bovine myocardium by radioligand binding
    • LOHSE, M.J., UKENA, D. & SCHWABE, U. (1985). Demonstration of Ri-type adenosine receptors in bovine myocardium by radioligand binding. Naunyn-Schmeideberg's Arch. Pharmacol., 328, 310-316.
    • (1985) Naunyn-Schmeideberg's Arch. Pharmacol. , vol.328 , pp. 310-316
    • Lohse, M.J.1    Ukena, D.2    Schwabe, U.3
  • 16
    • 0022399583 scopus 로고
    • Binding of agonists and antagonists to β-adrenoceptors in rat vas deferens: Relationship to functional response
    • MAY, J.M., ABEL, P.W. & MINNEMAN, K.P. (1985). Binding of agonists and antagonists to β-adrenoceptors in rat vas deferens: relationship to functional response. Naunyn-Schmiedeberg's Arch. Pharmacol., 331, 324-333.
    • (1985) Naunyn-Schmiedeberg's Arch. Pharmacol. , vol.331 , pp. 324-333
    • May, J.M.1    Abel, P.W.2    Minneman, K.P.3
  • 17
    • 0023265884 scopus 로고
    • Relationship between receptor occupancy and response at striatal dopamine autoreceptors
    • MELLER, E., BOHMAKER, K., NAMBA, Y., FRIEDHOFF, A.J. & GOLDSTEIN, M. (1987). Relationship between receptor occupancy and response at striatal dopamine autoreceptors. Mol. Pharmacol., 31, 592-598.
    • (1987) Mol. Pharmacol. , vol.31 , pp. 592-598
    • Meller, E.1    Bohmaker, K.2    Namba, Y.3    Friedhoff, A.J.4    Goldstein, M.5
  • 19
    • 0021336249 scopus 로고
    • 1-adrenergic receptors and the potency of agonist in rat vas deferens
    • 1-adrenergic receptors and the potency of agonist in rat vas deferens. Mol. Pharmacol., 25, 56-63.
    • (1984) Mol. Pharmacol. , vol.25 , pp. 56-63
    • Minneman, K.P.1    Abel, P.W.2
  • 21
    • 0025986796 scopus 로고
    • Characteristics of dose-dependent antagonism by B-funaltrexamine of the antinociceptive effect of intrathecal mu agonists
    • MJANGER, E. & YAKSH, T.L. (1991). Characteristics of dose-dependent antagonism by B-funaltrexamine of the antinociceptive effect of intrathecal mu agonists. J. Pharmacol. Exp. Ther., 258, 544-550.
    • (1991) J. Pharmacol. Exp. Ther. , vol.258 , pp. 544-550
    • Mjanger, E.1    Yaksh, T.L.2
  • 22
    • 0027213989 scopus 로고
    • Species comparison of adenosine and β-adrenoceptors in mammalian atrial and ventricular myocardium
    • MUSSER, B., MORGAN. M.E., LEID, M., MURRAY, T.F., LINDEN, J. & VESTRAL, R.E. (1993). Species comparison of adenosine and β-adrenoceptors in mammalian atrial and ventricular myocardium. Eur. J. Pharmacol., 246, 105-111.
    • (1993) Eur. J. Pharmacol. , vol.246 , pp. 105-111
    • Musser, B.1    Morgan, M.E.2    Leid, M.3    Murray, T.F.4    Linden, J.5    Vestral, R.E.6
  • 23
    • 0023510868 scopus 로고
    • 2-adrenergic receptor binding sites and the functional receptors inhibiting norepinephrine release in rat cerebral cortex
    • 2-adrenergic receptor binding sites and the functional receptors inhibiting norepinephrine release in rat cerebral cortex. J. Pharmacol. Exp. Ther., 32, 655-662.
    • (1987) J. Pharmacol. Exp. Ther. , vol.32 , pp. 655-662
    • Nasseri, A.1    Minneman, K.P.2
  • 24
    • 0026772582 scopus 로고
    • Development of tolerance to the analgesic activity of mu agonists after continuous infusion of morphine, meperidine or fentanyl in rats
    • PARONIS, C.A. & HOLTZMAN, S.G. (1992). Development of tolerance to the analgesic activity of mu agonists after continuous infusion of morphine, meperidine or fentanyl in rats. J. Pharmacol. Exp. Ther., 262, 1-9.
    • (1992) J. Pharmacol. Exp. Ther. , vol.262 , pp. 1-9
    • Paronis, C.A.1    Holtzman, S.G.2
  • 25
    • 0030435124 scopus 로고    scopus 로고
    • Electrophysiological effects of a novel, short-acting and potent ester derivative of amiodarone, ATI-2001, in guinea pig isolated heart
    • RAATIKAINEN, M.J.P., NAPOLITANO, C.A., DRUZGALA, P. & DENNIS, D.M. (1996). Electrophysiological effects of a novel, short-acting and potent ester derivative of amiodarone, ATI-2001, in guinea pig isolated heart. J. Pharmacol. Exp. Ther., 277, 1454-1463.
    • (1996) J. Pharmacol. Exp. Ther. , vol.277 , pp. 1454-1463
    • Raatikainen, M.J.P.1    Napolitano, C.A.2    Druzgala, P.3    Dennis, D.M.4
  • 28
    • 0029995339 scopus 로고    scopus 로고
    • 2D-adrenergic receptor regulation G protein activation in PC12 cell membranes
    • 2D-adrenergic receptor regulation G protein activation in PC12 cell membranes. Pharmacology, 52, 252-262.
    • (1996) Pharmacology , vol.52 , pp. 252-262
    • Tian, W.N.1    Duzic, E.2    Deth, R.C.3
  • 29
    • 0028831265 scopus 로고
    • Receptor reserve and affinity of mu opioid agonists in mouse antinociception: Correlation with receptor binding
    • ZERNIG, G., ISSAEVITCH, T., BROADBEAR, J.H., BURKE, T.F., LEWIS, J.W., BRINE, G.A. & WOODS, J.H. (1995). Receptor reserve and affinity of mu opioid agonists in mouse antinociception: Correlation with receptor binding. Life Sci., 57, 2113-2125.
    • (1995) Life Sci. , vol.57 , pp. 2113-2125
    • Zernig, G.1    Issaevitch, T.2    Broadbear, J.H.3    Burke, T.F.4    Lewis, J.W.5    Brine, G.A.6    Woods, J.H.7


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.