메뉴 건너뛰기




Volumn 50, Issue 1, 1996, Pages 196-205

A novel irreversible antagonist of the A1-adenosine receptor

Author keywords

[No Author keywords available]

Indexed keywords

2 [4 (2 CARBOXYETHYL)PHENETHYLAMINO]ADENOSINE 5' (N ETHYLCARBOXAMIDE); 8 CYCLOPENTYL 3 [3 [[4 (FLUOROSULFONYL)BENZOYL]OXY]PROPYL] 1 PROPYLXANTHINE; ADENOSINE A1 RECEPTOR; ADENOSINE A1 RECEPTOR ANTAGONIST; UNCLASSIFIED DRUG;

EID: 0030008733     PISSN: 0026895X     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article
Times cited : (27)

References (26)
  • 4
    • 0022268380 scopus 로고
    • 1 adenosine receptor: Identification of the binding subunit by photoaffinity crosslinking
    • 1 adenosine receptor: identification of the binding subunit by photoaffinity crosslinking. J. Biol. Chem. 260:10806-10811 (1985).
    • (1985) J. Biol. Chem. , vol.260 , pp. 10806-10811
    • Stiles, G.L.1    Daly, D.T.2    Olsson, R.A.3
  • 5
    • 0023009431 scopus 로고
    • 1 adenosine receptors: Persistent activation reveals spare receptors
    • 1 adenosine receptors: persistent activation reveals spare receptors. Mol. Pharmacol. 30:403-409 (1986).
    • (1986) Mol. Pharmacol. , vol.30 , pp. 403-409
    • Lohse, M.J.1    Klotz, K.2    Schwabe, U.3
  • 6
    • 0024205441 scopus 로고
    • 1 adenosine receptor: Identification of binding subunit
    • 1 adenosine receptor: identification of binding subunit. Mol. Pharmacol. 34:724-728 (1988).
    • (1988) Mol. Pharmacol. , vol.34 , pp. 724-728
    • Stiles, G.L.1    Jacobson, K.A.2
  • 10
    • 0020376510 scopus 로고
    • Calcium tolerant myocytes prepared by preincubation in a "KB medium."
    • Isenberg, G., and U. Klokner. Calcium tolerant myocytes prepared by preincubation in a "KB medium." Pfluegers Arch. 395:6-18 (1982).
    • (1982) Pfluegers Arch. , vol.395 , pp. 6-18
    • Isenberg, G.1    Klokner, U.2
  • 11
    • 0019441262 scopus 로고
    • Improved patch clamp techniques for high resolution current recordings from cells and cell-free membrane patches
    • Hamill, O. P., A. Marty, E. Neher, B. Sakmann, and F. J. Sigworth. Improved patch clamp techniques for high resolution current recordings from cells and cell-free membrane patches. Pfluegers Arch. 391:85-100 (1981).
    • (1981) Pfluegers Arch. , vol.391 , pp. 85-100
    • Hamill, O.P.1    Marty, A.2    Neher, E.3    Sakmann, B.4    Sigworth, F.J.5
  • 12
    • 0023936571 scopus 로고
    • Atrioventricular nodal accommodation in isolated guinea pig hearts: Physiological significance and role of adenosine
    • Jenkins, J., and L. Belardinelli. Atrioventricular nodal accommodation in isolated guinea pig hearts: physiological significance and role of adenosine. Circ. Res. 63:97-116 (1988).
    • (1988) Circ. Res. , vol.63 , pp. 97-116
    • Jenkins, J.1    Belardinelli, L.2
  • 13
    • 0023017977 scopus 로고
    • Effect of adenosine on atrioventricular conduction. I. Site and characterization of adenosine action in the guinea pig atrioventricular node
    • Clemo, H. F., and L. Belardinelli. Effect of adenosine on atrioventricular conduction. I. Site and characterization of adenosine action in the guinea pig atrioventricular node. Circ. Res. 59:427-436 (1986).
    • (1986) Circ. Res. , vol.59 , pp. 427-436
    • Clemo, H.F.1    Belardinelli, L.2
  • 14
    • 0022515173 scopus 로고
    • + channels by adenosine in isolated atrial myocytes: Involvement of GTP-binding proteins
    • + channels by adenosine in isolated atrial myocytes: involvement of GTP-binding proteins. Pfluegers Arch. 407:264-274 (1986).
    • (1986) Pfluegers Arch. , vol.407 , pp. 264-274
    • Kurachi, Y.1    Nakajima, T.2    Sugimoto, T.3
  • 15
    • 0021949426 scopus 로고
    • Covalent labeling of the β-adrenergic ligand binding site with para-(bromoacteamidyl)benzylcarazolol: A highly potent β-adrenergic affinity label
    • Dickinson, K. E., S. L. Heald, P. W. Jeffs, R. J. Lefkowitz, and M. G. Caron. Covalent labeling of the β-adrenergic ligand binding site with para-(bromoacteamidyl)benzylcarazolol: a highly potent β-adrenergic affinity label. Mol. Pharmacol. 27:499-506 (1985).
    • (1985) Mol. Pharmacol. , vol.27 , pp. 499-506
    • Dickinson, K.E.1    Heald, S.L.2    Jeffs, P.W.3    Lefkowitz, R.J.4    Caron, M.G.5
  • 18
    • 0026008320 scopus 로고
    • Evidence for impaired coupling of receptors to Gj protein in adipocytes from streptozocin-induced diabetic rats
    • Green, A., and J. L. Johnson. Evidence for impaired coupling of receptors to Gj protein in adipocytes from streptozocin-induced diabetic rats. Diabetes 40:88-94 (1991).
    • (1991) Diabetes , vol.40 , pp. 88-94
    • Green, A.1    Johnson, J.L.2
  • 21
    • 0028109356 scopus 로고
    • Novel approach for enhancing atrioventricular nodal conduction delay mediated by endogenous adenosine
    • Kollias-Baker, C., J. Xu, A. Pelleg, and L. Belardinelli. Novel approach for enhancing atrioventricular nodal conduction delay mediated by endogenous adenosine. Circ. Res. 75:972-980 (1994).
    • (1994) Circ. Res. , vol.75 , pp. 972-980
    • Kollias-Baker, C.1    Xu, J.2    Pelleg, A.3    Belardinelli, L.4
  • 22
    • 0025663017 scopus 로고
    • Drugs and receptors: An overview of the current state of knowledge
    • Kenakin, T. P. Drugs and receptors: an overview of the current state of knowledge. Drugs 40:666-687 (1991).
    • (1991) Drugs , vol.40 , pp. 666-687
    • Kenakin, T.P.1
  • 23
    • 0025305177 scopus 로고
    • Are molecular and electrophysiological data refining models of agonism?
    • Jenkinson, D., and A. Abbott. Are molecular and electrophysiological data refining models of agonism? Trends Pharmacol. Sci. 11:91-94 (1990).
    • (1990) Trends Pharmacol. Sci. , vol.11 , pp. 91-94
    • Jenkinson, D.1    Abbott, A.2
  • 24
    • 0022897429 scopus 로고
    • Differences in muscarinic receptor reserve for inhibition of adenylate cyclase and stimulation of phosphoinositide hydrolysis in chick heart cells
    • Brown, J. H., and D. Goldstein. Differences in muscarinic receptor reserve for inhibition of adenylate cyclase and stimulation of phosphoinositide hydrolysis in chick heart cells. Mol. Pharmacol. 30:466-470 (1986).
    • (1986) Mol. Pharmacol. , vol.30 , pp. 466-470
    • Brown, J.H.1    Goldstein, D.2
  • 25
    • 0023265884 scopus 로고
    • Relationship between receptor occupancy and response at striatal dopamine autoreceptors
    • Meller, E., K. Bohmaker, Y. Namba, A. J. Friedhoff, and M. Goldstein. Relationship between receptor occupancy and response at striatal dopamine autoreceptors. Mol. Pharmacol. 31:592-598 (1987).
    • (1987) Mol. Pharmacol. , vol.31 , pp. 592-598
    • Meller, E.1    Bohmaker, K.2    Namba, Y.3    Friedhoff, A.J.4    Goldstein, M.5
  • 26
    • 0002355204 scopus 로고
    • The use of haloalkylamines in the differentiation of receptors and the determination of dissociation constants of receptoragonist complexes
    • Furchgott, R. F. The use of haloalkylamines in the differentiation of receptors and the determination of dissociation constants of receptoragonist complexes. Adv. Drug. Res. 3:21-55 (1966).
    • (1966) Adv. Drug. Res. , vol.3 , pp. 21-55
    • Furchgott, R.F.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.