Metabolism and anti-HIV activity of phosphoramidate derivatives of D4T-MP with variations in the amino acid moiety

Advances in Experimental Medicine and Biology

Volumn 431, Issue , 1998, Pages 753-757

  Naesens, L ^a   Cahard, D ^b   Salgado, A ^b   Bidois, L ^b   De Clercq, E ^a   McGuigan, C ^b   Baizarini, J ^a  

^a REGA INSTITUTE FOR MEDICAL RESEARCH   (Belgium)

^b CARDIFF UNIVERSITY   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

ANTIVIRUS AGENT; STAVUDINE; STAVUDINE PHOSPHOROAMIDATE DERIVATIVE; THYMIDINE KINASE; UNCLASSIFIED DRUG;

AMINO ACID ANALYSIS; ANTIVIRAL ACTIVITY; CONFERENCE PAPER; DRUG ACTIVITY; DRUG EFFICACY; DRUG METABOLISM; ENZYME PHOSPHORYLATION; HUMAN; HUMAN CELL; HUMAN IMMUNODEFICIENCY VIRUS; PRIORITY JOURNAL; STRUCTURE ANALYSIS; VIRUS ACTIVATION;

AMINO ACIDS; ANIMALS; ANTI-HIV AGENTS; CELL LINE; CELL SURVIVAL; HIV-1; HIV-2; HUMANS; MICE; ORGANOPHOSPHORUS COMPOUNDS; PRODRUGS; STAVUDINE; STRUCTURE-ACTIVITY RELATIONSHIP; THYMIDINE KINASE;

CAVIA PORCELLUS; HUMAN IMMUNODEFICIENCY VIRUS; SUS SCROFA;

EID: 0031808057     PISSN: 00652598     EISSN: None     Source Type: Book Series    
DOI: 10.1007/978-1-4615-5381-6_144     Document Type: Article

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